SCHEMBL4251633

SCHEMBL4251633

COc1cc(N2Cc3ccc(Cl)cc3C2=O)ccc1N(C)C

nearest known ligand 0.58

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 12/20 0.58
HTR2A P28223 7/20 0.56
MCHR1 Q99705 4/20 0.45
HTR2B P41595 6/20 0.43
NPC1 O15118 1/20 0.41
PKM P14618 1/20 0.41
RAB9A P51151 1/20 0.41
CBLB Q13191 1/20 0.41
CYP3A4 P08684 1/20 0.41
CMA1 P23946 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4253666 0.91 HTR2C (0.58) HTR2CHTR2AMCHR1HTR2BNPC1
SCHEMBL4253075 0.87 NPC1 (0.47) HTR2CHTR2AMCHR1HTR2BNPC1
SCHEMBL4253350 0.86 NPC1 (0.48) HTR2CHTR2AMCHR1HTR2BNPC1
SCHEMBL4253635 0.84 NPC1 (0.60) HTR2CHTR2AMCHR1HTR2BNPC1
SCHEMBL4251879 0.80 NPC1 (0.45) HTR2CHTR2AMCHR1HTR2BNPC1
SCHEMBL4254603 0.80 NPC1 (0.51) HTR2CHTR2AMCHR1HTR2BNPC1
SCHEMBL4256261 0.79 HTR2C (0.44) HTR2CHTR2AMCHR1HTR2BNPC1
SCHEMBL4249678 0.79 CYP3A4 (0.47) HTR2CHTR2AMCHR1HTR2BNPC1
SCHEMBL4250602 0.79 HTR2C (0.47) HTR2CHTR2ANPC1PKMRAB9A
SCHEMBL4259106 0.78 CYP3A4 (0.43) MCHR1RAB9ACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009054653-A2 ISOINDOLONES WITH HIGH BINDING AFFINITY TO BETA-AMYLOID AGGREGATES AND FIBRILS, AND ITS USE AND PREPARATION METHOD KOREA INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 2009-04-30 WO claimed
WO-2009054653-A2 ISOINDOLONES WITH HIGH BINDING AFFINITY TO BETA-AMYLOID AGGREGATES AND FIBRILS, AND ITS USE AND PREPARATION METHOD KOREA INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 2009-04-30 WO disclosed