SCHEMBL4249678

SCHEMBL4249678

COc1cc(N2Cc3cc(F)ccc3C2=O)ccc1N(C)C

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.47
UGCG Q16739 2/20 0.47
NPC1 O15118 2/20 0.46
RAB9A P51151 2/20 0.46
HTR2C P28335 8/20 0.44
PKM P14618 1/20 0.41
PIK3CG P48736 3/20 0.41
HTR2A P28223 3/20 0.39
HTR2B P41595 3/20 0.39
MCHR1 Q99705 2/20 0.39
DRD2 P14416 1/20 0.38
DRD4 P21917 1/20 0.38
DRD3 P35462 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4253350 0.91 NPC1 (0.48) CYP3A4UGCGNPC1RAB9AHTR2C
SCHEMBL4254603 0.87 NPC1 (0.51) CYP3A4NPC1RAB9AHTR2CPKM
SCHEMBL4251879 0.87 NPC1 (0.45) CYP3A4UGCGNPC1RAB9AHTR2C
SCHEMBL4253666 0.86 HTR2C (0.58) CYP3A4NPC1RAB9AHTR2CPKM
SCHEMBL4256261 0.86 HTR2C (0.44) CYP3A4NPC1RAB9AHTR2CPKM
SCHEMBL4253635 0.84 NPC1 (0.60) CYP3A4UGCGNPC1RAB9AHTR2C
SCHEMBL4253075 0.80 NPC1 (0.47) UGCGNPC1RAB9AHTR2CPKM
SCHEMBL4251633 0.79 HTR2C (0.58) CYP3A4NPC1RAB9AHTR2CPKM
SCHEMBL4258064 0.79 PARP1 (0.46) CYP3A4UGCGNPC1RAB9APKM
SCHEMBL4250037 0.78 CYP3A4 (0.50) CYP3A4RAB9AMCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009054653-A2 ISOINDOLONES WITH HIGH BINDING AFFINITY TO BETA-AMYLOID AGGREGATES AND FIBRILS, AND ITS USE AND PREPARATION METHOD KOREA INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 2009-04-30 WO disclosed