SCHEMBL4256261

SCHEMBL4256261

COc1cc(N2Cc3cc(Br)ccc3C2=O)ccc1N(C)C

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 8/20 0.44
BACE1 P56817 1/20 0.43
NPC1 O15118 7/20 0.41
RAB9A P51151 7/20 0.41
PKM P14618 2/20 0.41
PIK3CG P48736 2/20 0.41
HTR2A P28223 4/20 0.39
HTR2B P41595 3/20 0.39
MCHR1 Q99705 1/20 0.39
CYP3A4 P08684 1/20 0.37
POLB P06746 1/20 0.36
TP53 P04637 1/20 0.36
GAA P10253 1/20 0.36
TSHR P16473 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4254603 0.87 NPC1 (0.51) HTR2CNPC1RAB9APKMPIK3CG
SCHEMBL4251879 0.87 NPC1 (0.45) HTR2CNPC1RAB9APKMPIK3CG
SCHEMBL4249678 0.86 CYP3A4 (0.47) HTR2CNPC1RAB9APKMPIK3CG
SCHEMBL4253666 0.86 HTR2C (0.58) HTR2CNPC1RAB9APKMPIK3CG
SCHEMBL4253635 0.84 NPC1 (0.60) HTR2CNPC1RAB9APKMPIK3CG
SCHEMBL4253075 0.80 NPC1 (0.47) HTR2CNPC1RAB9APKMHTR2A
SCHEMBL4253350 0.79 NPC1 (0.48) HTR2CNPC1RAB9APKMHTR2A
SCHEMBL4251633 0.79 HTR2C (0.58) HTR2CNPC1RAB9APKMHTR2A
SCHEMBL4251115 0.79 PARP1 (0.46) BACE1NPC1RAB9APKMCYP3A4
SCHEMBL4253067 0.78 ESR1 (0.52) RAB9AMCHR1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009054653-A2 ISOINDOLONES WITH HIGH BINDING AFFINITY TO BETA-AMYLOID AGGREGATES AND FIBRILS, AND ITS USE AND PREPARATION METHOD KOREA INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 2009-04-30 WO claimed
WO-2009054653-A2 ISOINDOLONES WITH HIGH BINDING AFFINITY TO BETA-AMYLOID AGGREGATES AND FIBRILS, AND ITS USE AND PREPARATION METHOD KOREA INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 2009-04-30 WO disclosed