SCHEMBL4251963

SCHEMBL4251963

Cc1ccc(CN(Cc2ccccc2)C(CCN(Cc2ccccc2)C(=O)O)Cc2cncs2)s1

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 14/20 0.37
CYP2D6 P10635 3/20 0.37
FNTA P49354 1/20 0.34
FNTB P49356 1/20 0.34
CYP2C9 P11712 2/20 0.34
CYP2C19 P33261 2/20 0.34
GPR142 Q7Z601 3/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
POLB P06746 1/20 0.33
GAA P10253 1/20 0.33
MAPT P10636 1/20 0.33
PKM P14618 1/20 0.33
HPGD P15428 1/20 0.33
RECQL P46063 1/20 0.33
BLM P54132 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4253307 0.80 GPR142 (0.37) CYP3A4GPR142
SCHEMBL893625 0.71 CYP3A4 (0.51) CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL4245373 0.68 CYP3A4 (0.38) CYP3A4CYP2D6CYP2C9CYP2C19ALDH1A1
SCHEMBL4248044 0.66 CYP3A4 (0.57) CYP3A4CYP2D6CYP2C9CYP2C19LMNA
SCHEMBL13780920 0.65 CYP3A4 (0.61) CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL9944032 0.65 CYP3A4 (0.49) CYP3A4GPR142
SCHEMBL893063 0.63 CYP3A4 (0.59) CYP3A4CYP2D6CYP2C9CYP2C19LMNA
SCHEMBL893562 0.63 CYP3A4 (0.51) CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL4255741 0.61 NPSR1 (0.37) CYP3A4CYP2D6CYP2C9CYP2C19ALDH1A1
SCHEMBL893483 0.61 TDP1 (0.50) CYP3A4CYP2D6CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2081917-A2 CYTOCHROME P450 OXIDASE INHIBITORS AND USES THEREOF Abbott Laboratories (US) 2009-07-29 EP disclosed
WO-2008027932-A2 CYTOCHROME P450 OXIDASE INHIBITORS AND USES THEREOF ABBOTT LABORATORIES (US) 2008-03-06 WO disclosed