SCHEMBL4255741

SCHEMBL4255741

[CH](Cc1ccccc1)CC(Cc1cncs1)N(Cc1ccccc1)Cc1ccco1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 9/20 0.37
MAPT P10636 7/20 0.37
ALDH1A1 P00352 6/20 0.37
TSHR P16473 4/20 0.37
HTT P42858 4/20 0.37
LMNA P02545 3/20 0.37
USP2 O75604 2/20 0.37
CYP3A4 P08684 2/20 0.37
CYP2C9 P11712 2/20 0.37
CYP2C19 P33261 2/20 0.37
CYP2D6 P10635 1/20 0.37
KDM4E B2RXH2 4/20 0.36
MEN1 O00255 4/20 0.35
KMT2A Q03164 4/20 0.35
HSD17B10 Q99714 3/20 0.35
L3MBTL1 Q9Y468 2/20 0.35
ALOX15 P16050 1/20 0.35
CASP1 P29466 1/20 0.35
TP53 P04637 3/20 0.34
MAPK1 P28482 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4255744 0.65 MAPT (0.35) NPSR1MAPTALDH1A1TSHRHTT
SCHEMBL4251963 0.61 CYP3A4 (0.37) MAPTALDH1A1LMNACYP3A4CYP2C9
SCHEMBL9389496 0.58 SLC6A3 (0.49) LMNATDP1
Furfenorex SCHEMBL164756 0.58 ADRA2B (0.65) NPSR1MAPTALDH1A1TSHRHTT
SCHEMBL16523570 0.58 TSHR (0.51) NPSR1MAPTALDH1A1TSHRHTT
SCHEMBL27825512 0.57 SLC6A3 (0.47) TDP1
SCHEMBL5790031 0.57 TSHR (0.52) NPSR1MAPTALDH1A1TSHRHTT
SCHEMBL28141333 0.57 TSHR (0.54) TSHRLMNACYP3A4KDM4EPOLB
SCHEMBL7471615 0.57 LMNA (0.38) ALDH1A1TSHRHTTLMNAUSP2
SCHEMBL7040606 0.56 SLC6A3 (0.54)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2081917-A2 CYTOCHROME P450 OXIDASE INHIBITORS AND USES THEREOF Abbott Laboratories (US) 2009-07-29 EP claimed
WO-2008027932-A2 CYTOCHROME P450 OXIDASE INHIBITORS AND USES THEREOF ABBOTT LABORATORIES (US) 2008-03-06 WO claimed
EP-2081917-A2 CYTOCHROME P450 OXIDASE INHIBITORS AND USES THEREOF Abbott Laboratories (US) 2009-07-29 EP disclosed
WO-2008027932-A2 CYTOCHROME P450 OXIDASE INHIBITORS AND USES THEREOF ABBOTT LABORATORIES (US) 2008-03-06 WO disclosed