SCHEMBL4252371

SCHEMBL4252371

CCCCOC(=O)c1c(C=CC(=O)O)cccc1C(F)(F)F

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
TP53 P04637 1/20 0.44
L3MBTL1 Q9Y468 3/20 0.42
LMNA P02545 2/20 0.42
ALDH1A1 P00352 2/20 0.42
TSHR P16473 2/20 0.42
TDP1 Q9NUW8 2/20 0.42
KDM4E B2RXH2 1/20 0.42
MAOB P27338 4/20 0.41
NFKB1 P19838 1/20 0.41
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
HCAR2 Q8TDS4 1/20 0.40
ESR1 P03372 1/20 0.39
PLK1 P53350 1/20 0.39
PLK3 Q9H4B4 1/20 0.39
CYP3A4 P08684 1/20 0.39
MAPK1 P28482 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4243404 0.79 MAOB (0.46) MAPTSMN1; SMN2LMNAKDM4EMAOB
SCHEMBL4243406 0.79 MAOB (0.46) MAPTSMN1; SMN2LMNAKDM4EMAOB
SCHEMBL4473051 0.78 MAOB (0.45) MAPTSMN1; SMN2LMNAKDM4EMAOB
SCHEMBL4473057 0.78 MAOB (0.45) MAPTSMN1; SMN2LMNAKDM4EMAOB
SCHEMBL9518819 0.73 NFKB1 (0.50) MAPTSMN1; SMN2LMNAKDM4EMAOB
SCHEMBL10984242 0.73 BACE1 (0.56) MAPTSMN1; SMN2LMNAMAOBNFKB1
SCHEMBL28299341 0.72 TSHR (0.71) TP53L3MBTL1LMNAALDH1A1TSHR
SCHEMBL4469618 0.70 LMNA (0.49) MAPTLMNAALDH1A1MAOBNFKB1
SCHEMBL4469625 0.70 LMNA (0.49) MAPTLMNAALDH1A1MAOBNFKB1
SCHEMBL4469622 0.70 LMNA (0.49) MAPTLMNAALDH1A1MAOBNFKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1773833-A4 PYRROLO(OXO)QUINOLINES AS 5HT LIGANDS BRISTOL MYERS SQUIBB CO (US) 2009-07-22 EP disclosed
EP-1773833-A2 PYRROLO(OXO)QUINOLINES AS 5HT LIGANDS Bristol-Myers Squibb Company (US) 2007-04-18 EP disclosed
WO-2006019940-A2 PYRROLO(OXO)QUINOLINES AS 5HT LIGANDS BRISTOL-MYERS SQUIBB COMPANY (US) 2006-02-23 WO disclosed