SCHEMBL4254039

SCHEMBL4254039

COc1ccc2c(c1)C(=O)N(c1ccc([N+](=O)[O-])cc1)C2=O

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN2A Q99250 1/20 0.61
ESR1 P03372 1/20 0.58
CA12 O43570 2/20 0.56
CA9 Q16790 2/20 0.56
CA1 P00915 1/20 0.56
CA2 P00918 1/20 0.56
LPAR1 Q92633 1/20 0.52
LPAR5 Q9H1C0 1/20 0.52
LPAR3 Q9UBY5 1/20 0.52
MEN1 O00255 6/20 0.51
KMT2A Q03164 6/20 0.51
ALDH1A1 P00352 2/20 0.51
MAPT P10636 2/20 0.51
HTT P42858 2/20 0.49
KDM4E B2RXH2 1/20 0.49
LMNA P02545 1/20 0.49
GAA P10253 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
PTPN7 P35236 1/20 0.48
PTPN22 Q9Y2R2 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11689784 0.83 CA12 (0.67) SCN2ACA12CA9CA1CA2
SCHEMBL11724682 0.82 ALDH1A1 (0.53) ESR1CA12KMT2AALDH1A1MAPT
SCHEMBL11724665 0.82 KMT2A (0.52) SCN2AESR1CA12MEN1KMT2A
SCHEMBL4255804 0.80 ESR1 (0.64) SCN2AESR1CA12CA9CA1
SCHEMBL28911652 0.80 CA12 (0.70) SCN2ACA12CA9CA1CA2
SCHEMBL10013240 0.79 ALDH1A1 (0.65) SCN2AESR1CA9CA1MEN1
SCHEMBL12639212 0.79 ESR1 (0.72) ESR1MEN1KMT2AALDH1A1MAPT
SCHEMBL17326265 0.78 SCN2A (0.67) SCN2AESR1CA12CA9CA1
SCHEMBL4251148 0.77 NPC1 (0.58) ESR1CA9CA1CA2MEN1
SCHEMBL4258439 0.77 ESR1 (0.61) ESR1CA12CA9CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009054653-A2 ISOINDOLONES WITH HIGH BINDING AFFINITY TO BETA-AMYLOID AGGREGATES AND FIBRILS, AND ITS USE AND PREPARATION METHOD KOREA INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 2009-04-30 WO disclosed