SCHEMBL4255804

SCHEMBL4255804

COc1ccc2c(c1)C(=O)N(c1ccc(N)cc1)C2=O

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.64
ALDH1A1 P00352 4/20 0.62
NPC1 O15118 3/20 0.62
RAB9A P51151 3/20 0.62
TSHR P16473 2/20 0.62
CASP1 P29466 2/20 0.62
CASP7 P55210 1/20 0.62
HSD17B10 Q99714 1/20 0.62
MEN1 O00255 6/20 0.56
KMT2A Q03164 6/20 0.56
MAPK1 P28482 1/20 0.54
NPSR1 Q6W5P4 1/20 0.54
GAA P10253 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
HTT P42858 1/20 0.53
NR1H3 Q13133 2/20 0.52
SCN2A Q99250 1/20 0.52
KDM4E B2RXH2 1/20 0.51
NR1H2 P55055 1/20 0.50
BRD4 O60885 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21082652 0.87 BRD4 (0.64) ESR1ALDH1A1NPC1RAB9ATSHR
SCHEMBL21082653 0.86 BRD4 (0.62) ESR1ALDH1A1NPC1RAB9ATSHR
SCHEMBL12639212 0.84 ESR1 (0.72) ESR1ALDH1A1RAB9AMEN1KMT2A
SCHEMBL10013240 0.84 ALDH1A1 (0.65) ESR1ALDH1A1MEN1KMT2AGAA
SCHEMBL4258275 0.82 ESR1 (0.61) ESR1ALDH1A1MEN1KMT2ANPSR1
SCHEMBL4258439 0.82 ESR1 (0.61) ESR1ALDH1A1MEN1KMT2AMAPK1
SCHEMBL9566650 0.81 CASP1 (0.83) ESR1ALDH1A1NPC1RAB9ATSHR
SCHEMBL12639223 0.81 ESR1 (0.72) ESR1ALDH1A1MEN1KMT2AHTT
SCHEMBL9468586 0.81 ALDH1A1 (0.71) ESR1ALDH1A1NPC1RAB9ATSHR
SCHEMBL12898395 0.81 ESR1 (0.59) ESR1ALDH1A1RAB9AMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009054653-A2 ISOINDOLONES WITH HIGH BINDING AFFINITY TO BETA-AMYLOID AGGREGATES AND FIBRILS, AND ITS USE AND PREPARATION METHOD KOREA INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 2009-04-30 WO claimed
WO-2009054653-A2 ISOINDOLONES WITH HIGH BINDING AFFINITY TO BETA-AMYLOID AGGREGATES AND FIBRILS, AND ITS USE AND PREPARATION METHOD KOREA INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 2009-04-30 WO disclosed