SCHEMBL4255208

SCHEMBL4255208

CP(=O)(O)CCCC(=O)O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 6/20 0.52
GABBR2 O75899 1/20 0.52
CYP1A2 P05177 1/20 0.52
THPO P40225 1/20 0.52
GABBR1 Q9UBS5 1/20 0.52
LMNA P02545 3/20 0.50
BLM P54132 1/20 0.50
SLC22A6 Q4U2R8 2/20 0.48
NFKB1 P19838 1/20 0.46
PMP22 Q01453 1/20 0.46
AKR1B1 P15121 1/20 0.44
ALDH1A1 P00352 3/20 0.43
PPARG P37231 6/20 0.42
PPARD Q03181 6/20 0.42
PPARA Q07869 6/20 0.42
GPR84 Q9NQS5 5/20 0.42
HDAC11 Q96DB2 5/20 0.42
TLR2 O60603 2/20 0.42
TDP1 Q9NUW8 2/20 0.42
FABP4 P15090 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16104630 0.84
SCHEMBL63051 0.84
SCHEMBL28187226 0.82 TSHR (0.42) TSHRGABBR2CYP1A2THPOGABBR1
Hydrochloric Acid SCHEMBL11709036 0.82 LMNA (0.46) TSHRGABBR2CYP1A2THPOGABBR1
SCHEMBL5554876 0.82 TSHR (0.42) TSHRGABBR2CYP1A2THPOGABBR1
SCHEMBL28186481 0.82 TSHR (0.42) TSHRGABBR2CYP1A2THPOGABBR1
SCHEMBL6037799 0.80 FOLH1 (0.61)
SCHEMBL307497 0.79 TYMS (0.58) TSHRLMNABLMSLC22A6NFKB1
SCHEMBL11287065 0.78 GABBR2 (0.68) TSHRGABBR2CYP1A2THPOGABBR1
SCHEMBL11347827 0.78 GABBR2 (0.68) TSHRGABBR2CYP1A2THPOGABBR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 41 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116390925-A AMPK activator 卡尔优普公司 2023-07-04 CN claimed
EP-3956336-A1 METHODS FOR PRODUCING CRYSTALLINE L-GLUFOSINATE AMMONIUM MONOHYDRATE BASF SE (DE) 2022-02-23 EP claimed
WO-2020214631-A1 METHODS FOR PRODUCING CRYSTALLINE L-GLUFOSINATE AMMONIUM MONOHYDRATE AGRIMETIS, LLC (US) 2020-10-22 WO claimed
EP-1752143-A1 Novel uses for drugs targeting glutamine synthetase NewThera (FR) 2007-02-14 EP claimed
WO-2025061721-A1 HERBICIDAL COMPOSITIONS COMPRISING SPECIFIC SURFACTANTS SPECIALTY OPERATIONS FRANCE (FR) 2025-03-27 WO disclosed
WO-2024069167-A1 AN HERBICIDAL COMBINATION, COMPOSITION AND METHOD OF CONTROLLING WEEDS USING THE SAME UPL MAURITIUS LIMITED (MU) 2024-04-04 WO disclosed
EP-4314310-A1 METHODS FOR PREPARING L-GLUFOSINATE BASF SE (DE) 2024-02-07 EP disclosed
CN-116390925-A AMPK activator 卡尔优普公司 2023-07-04 CN disclosed
WO-2022207753-A1 METHODS FOR PREPARING L-GLUFOSINATE BASF SE (DE) 2022-10-06 WO disclosed
EP-3956336-A1 METHODS FOR PRODUCING CRYSTALLINE L-GLUFOSINATE AMMONIUM MONOHYDRATE BASF SE (DE) 2022-02-23 EP disclosed
EP-3847269-A1 METHODS FOR IMPROVING YIELDS OF L-GLUFOSINATE BASF SE (DE) 2021-07-14 EP disclosed
WO-2020214631-A1 METHODS FOR PRODUCING CRYSTALLINE L-GLUFOSINATE AMMONIUM MONOHYDRATE AGRIMETIS, LLC (US) 2020-10-22 WO disclosed
EP-1752143-A1 Novel uses for drugs targeting glutamine synthetase NewThera (FR) 2007-02-14 EP disclosed
WO-1998048611-A9 CROP HETEROSIS AND HERBICIDE YAN WENGUI (US) 1999-03-25 WO disclosed
EP-0402769-A1 Liquid herbicidal mixture formulations HOECHST AKTIENGESELLSCHAFT (DE) 1990-12-19 EP disclosed
US-4960928-A 1-Hydroxy-omega-(alkyl- or arylphosphinico)alkane-1,1-diphosphonic acids, salts thereof, and processes for the preparation of these compounds Hoechst Aktiengesellschaft Knapsack (DE) 1990-10-02 US disclosed
EP-0358428-A2 Process for producing optically active compounds NISSAN CHEMICAL INDUSTRIES, LIMITED (JP) 1990-03-14 EP disclosed
EP-0330022-A2 1-Hydroxy-omega-(alkyl- or arylphosphinico-)alkane-1,1-diphosphonic acids, their salts and process for preparing these compounds HOECHST AKTIENGESELLSCHAFT (DE) 1989-08-30 EP disclosed
EP-0249188-A2 Process for the production of L-2-amino-4-(hydroxymethyl-phosphinyl)-butyric acid MEIJI SEIKA KAISHA LTD. (JP) 1987-12-16 EP disclosed
EP-0018415-B1 PROCESS FOR PRODUCING ALKYL 4-(ALKOXY METHYL PHOSPHINOYL)BUTYRATES AND ALKYL-(2-AMINO-4-(ALKOXY METHYL PHOSPHINOYL)) BUTYRATES MEIJI SEIKA KAISHA LTD. (JP) 1982-10-13 EP disclosed