SCHEMBL4256175

SCHEMBL4256175

Cc1cc(CNCCC(C)C)ccc1-c1ccc(-c2nnc[nH]2)cc1

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 1/20 0.38
S1PR1 P21453 1/20 0.35
VSIR Q9H7M9 5/20 0.34
HDAC1 Q13547 1/20 0.33
MAPT P10636 1/20 0.32
MAPK1 P28482 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
CD274 Q9NZQ7 2/20 0.32
PDCD1 Q15116 1/20 0.32
OPRL1 P41146 1/20 0.31
NSD2 O96028 1/20 0.31
MAPK14 Q16539 2/20 0.31
ITGB1 P05556 1/20 0.30
ITGA4 P13612 1/20 0.30
ITGB7 P26010 1/20 0.30
ALDH2 P05091 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4082823 0.93 AKT1 (0.39) AKT1S1PR1VSIRHDAC1CD274
SCHEMBL4074510 0.90 AKT1 (0.36) AKT1VSIRHDAC1MAPTMAPK1
SCHEMBL4081718 0.88 AKT1 (0.35) AKT1S1PR1VSIRHDAC1MAPT
SCHEMBL4080115 0.88 AKT1 (0.35) AKT1S1PR1VSIRHDAC1OPRL1
SCHEMBL4071465 0.79 CSNK2A1 (0.40) AKT1VSIRHDAC1CD274OPRL1
SCHEMBL13633146 0.79 SCN8A (0.35) AKT1S1PR1VSIRHDAC1CD274
Hydrochloric Acid SCHEMBL4490670 0.78 SCN8A (0.35) AKT1S1PR1VSIRHDAC1CD274
SCHEMBL13137130 0.77 HTT (0.39) AKT1S1PR1VSIRHDAC1MAPT
Hydrochloric Acid SCHEMBL3050316 0.76 HTT (0.39) AKT1S1PR1VSIRHDAC1MAPT
SCHEMBL4081754 0.73 KDM4E (0.41) HDAC1MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2084127-A1 DIARYL, DIPYRIDINYL AND ARYL-PYRIDINYL DERIVATIVES AND USES THEREOF Pfizer Products Inc. (US) 2009-08-05 EP claimed
WO-2008059335-A1 DIARYL, DIPYRIDINYL AND ARYL-PYRIDINYL DERIVATIVES AND USES THEREOF PFIZER PRODUCTS INC. (US) 2008-05-22 WO claimed