SCHEMBL4074510

SCHEMBL4074510

Cc1cc(CNCCC(C)C)ccc1-c1cccc(-c2nnc[nH]2)c1

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 1/20 0.36
VSIR Q9H7M9 8/20 0.36
ALDH2 P05091 1/20 0.34
HDAC1 Q13547 1/20 0.34
CD274 Q9NZQ7 6/20 0.32
PDCD1 Q15116 5/20 0.32
SCN8A Q9UQD0 1/20 0.32
CA2 P00918 1/20 0.31
MAPT P10636 1/20 0.30
MAPK1 P28482 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4256175 0.90 AKT1 (0.38) AKT1VSIRALDH2HDAC1CD274
SCHEMBL13633146 0.89 SCN8A (0.35) AKT1VSIRHDAC1CD274SCN8A
SCHEMBL4071465 0.89 CSNK2A1 (0.40) AKT1VSIRHDAC1CD274CA2
SCHEMBL4082823 0.88 AKT1 (0.39) AKT1VSIRHDAC1CD274PDCD1
Hydrochloric Acid SCHEMBL4490670 0.88 SCN8A (0.35) AKT1VSIRHDAC1CD274SCN8A
SCHEMBL4080115 0.85 AKT1 (0.35) AKT1VSIRHDAC1SCN8A
SCHEMBL4083648 0.81 HDAC1 (0.33) AKT1VSIRHDAC1CA2
SCHEMBL4081718 0.79 AKT1 (0.35) AKT1VSIRHDAC1CD274MAPT
SCHEMBL1347921 0.75 OPRM1 (0.46) ALDH2HDAC1CD274PDCD1CA2
SCHEMBL13137130 0.74 HTT (0.39) AKT1VSIRALDH2HDAC1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2084127-A1 DIARYL, DIPYRIDINYL AND ARYL-PYRIDINYL DERIVATIVES AND USES THEREOF Pfizer Products Inc. (US) 2009-08-05 EP claimed
WO-2008059335-A1 DIARYL, DIPYRIDINYL AND ARYL-PYRIDINYL DERIVATIVES AND USES THEREOF PFIZER PRODUCTS INC. (US) 2008-05-22 WO claimed