SCHEMBL4081718

SCHEMBL4081718

CC(C)CCNCc1ccc(-c2ccc(-c3nnc[nH]3)cc2)c(F)c1

nearest known ligand 0.35

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 1/20 0.35
HDAC1 Q13547 1/20 0.33
PDCD1LG2 Q9BQ51 1/20 0.32
CD274 Q9NZQ7 1/20 0.32
S1PR1 P21453 1/20 0.32
VSIR Q9H7M9 2/20 0.32
MAPK14 Q16539 1/20 0.32
MAPT P10636 1/20 0.31
MAPK1 P28482 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
BACE1 P56817 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13633146 0.91 SCN8A (0.35) AKT1HDAC1PDCD1LG2CD274S1PR1
Hydrochloric Acid SCHEMBL4490670 0.90 SCN8A (0.35) AKT1HDAC1PDCD1LG2CD274S1PR1
SCHEMBL4256175 0.88 AKT1 (0.38) AKT1HDAC1CD274S1PR1VSIR
SCHEMBL4080115 0.85 AKT1 (0.35) AKT1HDAC1S1PR1VSIRMAPK14
SCHEMBL4082823 0.83 AKT1 (0.39) AKT1HDAC1CD274S1PR1VSIR
SCHEMBL4083648 0.80 HDAC1 (0.33) AKT1HDAC1VSIR
SCHEMBL4074510 0.79 AKT1 (0.36) AKT1HDAC1CD274VSIRMAPT
SCHEMBL4071465 0.78 CSNK2A1 (0.40) AKT1HDAC1PDCD1LG2CD274VSIR
SCHEMBL30312213 0.71 DHODH (0.41)
SCHEMBL13633142 0.70 OPRM1 (0.45) HDAC1S1PR1BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2084127-A1 DIARYL, DIPYRIDINYL AND ARYL-PYRIDINYL DERIVATIVES AND USES THEREOF Pfizer Products Inc. (US) 2009-08-05 EP claimed
WO-2008059335-A1 DIARYL, DIPYRIDINYL AND ARYL-PYRIDINYL DERIVATIVES AND USES THEREOF PFIZER PRODUCTS INC. (US) 2008-05-22 WO claimed