SCHEMBL4257003

SCHEMBL4257003

O=C1Oc2ccc(O)cc2C1=Cc1ccc(O)c(O)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TOP1 P11387 3/20 1.00
STK17B O94768 4/20 0.67
TOP2A P11388 1/20 0.56
MEN1 O00255 4/20 0.56
KMT2A Q03164 4/20 0.56
RECQL P46063 3/20 0.56
AURKA O14965 3/20 0.56
GSK3B P49841 3/20 0.56
CDK5 Q00535 3/20 0.56
DAPK3 O43293 2/20 0.56
BLK P51451 2/20 0.56
TEK Q02763 2/20 0.56
BTK Q06187 2/20 0.56
ITK Q08881 2/20 0.56
STK17A Q9UEE5 2/20 0.56
DAPK2 Q9UIK4 2/20 0.56
CDK5R1 Q15078 2/20 0.56
MAOA P21397 2/20 0.56
KDM4E B2RXH2 1/20 0.56
PSMD14 O00487 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4256999 1.00 TOP1 (1.00) TOP1STK17BTOP2AMEN1KMT2A
SCHEMBL29406646 0.88 TOP1 (0.78) TOP1STK17BTOP2AMEN1KMT2A
SCHEMBL4267530 0.85 TOP1 (0.76) TOP1STK17BTOP2AMEN1KMT2A
SCHEMBL4267528 0.85 TOP1 (0.76) TOP1STK17BTOP2AMEN1KMT2A
SCHEMBL4264851 0.84 TOP1 (0.73) TOP1STK17BMEN1KMT2ARECQL
SCHEMBL4264849 0.84 TOP1 (0.73) TOP1STK17BMEN1KMT2ARECQL
SCHEMBL30337058 0.80 STK17B (1.00) TOP1STK17BMEN1KMT2ARECQL
Isoaurostatin SCHEMBL15426107 0.76 MAOA (0.63) TOP1STK17BTOP2AMEN1KMT2A
Isoaurostatin SCHEMBL29551912 0.76 MAOA (0.63) TOP1STK17BTOP2AMEN1KMT2A
SCHEMBL3676919 0.76 TOP1 (0.70) TOP1TOP2AGAAEGFRIGF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7629375-B2 Cytoprotective compounds, pharmaceutical and cosmetic formulations, and methods JOHNSON & JOHNSON CONSUMER COMPANIES, INC. (US) 2009-12-08 US disclosed
US-20060178356-A1 Cytoprotective compounds, pharmaceutical and cosmetic formulations, and methods GALILEO PHARMACEUTICALS, INC. 2006-08-10 US disclosed
EP-1435894-A4 CYTOPROTECTIVE COMPOUNDS, PHARMACEUTICAL AND COSMETIC FORMULATIONS, AND METHODS GALILEO PHARMACEUTICALS INC (US) 2005-07-06 EP disclosed
US-20050142155-A1 Cytoprotective compounds, pharmaceutical and cosmetic formulations, and methods JOHNSON & JOHNSON CONSUMER INC. 2005-06-30 US disclosed
US-20050113416-A1 Cytoprotective compounds, pharmaceutical and cosmetic formulations, and methods GALILEO PHARMACEUTICALS, INC. 2005-05-26 US disclosed
EP-1435894-A2 CYTOPROTECTIVE COMPOUNDS, PHARMACEUTICAL AND COSMETIC FORMULATIONS, AND METHODS Galileo Pharmaceuticals, Inc. (US) 2004-07-14 EP disclosed
US-20030073712-A1 Cytoprotective compounds, pharmaceutical and cosmetic formulations, and methods JOHNSON & JOHNSON CONSUMER COMPANIES, INC. 2003-04-17 US disclosed
WO-2003009807-A2 CYTOPROTECTIVE COMPOUNDS, PHARMACEUTICAL AND COSMETIC FORMULATIONS, AND METHODS GALILEO LABORATORIES, INC. (US) 2003-02-06 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050142155-A1 Cytoprotective compounds, pharmaceutical and cosmetic formulations, and methods HSF1, HMOX1, NQO1 TOP1 1758/4885STK17B 2724/4885TOP2A 1419/4885
US-20030073712-A1 Cytoprotective compounds, pharmaceutical and cosmetic formulations, and methods HSF1, HMOX1, NQO1 TOP1 1758/4885STK17B 2724/4885TOP2A 1419/4885
US-20050113416-A1 Cytoprotective compounds, pharmaceutical and cosmetic formulations, and methods HSF1, HMOX1, NQO1 TOP1 1758/4885STK17B 2724/4885TOP2A 1419/4885
US-20060178356-A1 Cytoprotective compounds, pharmaceutical and cosmetic formulations, and methods HSF1, HMOX1, NQO1 TOP1 1758/4885STK17B 2724/4885TOP2A 1419/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.