SCHEMBL4257883

SCHEMBL4257883

Cc1cccn2c(-c3nc(N[C@@H](C)c4ccc(Br)cc4)ncc3C#N)cnc12

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.43
HPGD P15428 2/20 0.43
KDM4E B2RXH2 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
PLK1 P53350 4/20 0.39
RPS6KB1 P23443 1/20 0.34
KDR P35968 3/20 0.34
CDK1 P06493 2/20 0.34
IGF1R P08069 3/20 0.33
ELANE P08246 1/20 0.33
CTRB1 P17538 1/20 0.33
CDK2 P24941 1/20 0.33
AR P10275 1/20 0.32
IDH1 O75874 5/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3546850 0.92 PLK1 (0.47) ALDH1A1HPGDSMN1; SMN2PLK1RPS6KB1
SCHEMBL3546619 0.91 PLK1 (0.39) ALDH1A1HPGDKDM4ESMN1; SMN2PLK1
SCHEMBL3558617 0.91 PLK1 (0.39) ALDH1A1HPGDKDM4ESMN1; SMN2PLK1
SCHEMBL3550499 0.91 PLK1 (0.39) PLK1RPS6KB1AR
SCHEMBL3552091 0.88 PLK1 (0.38) ALDH1A1HPGDKDM4EPLK1RPS6KB1
SCHEMBL3558801 0.88 PLK1 (0.38) ALDH1A1HPGDKDM4EPLK1RPS6KB1
SCHEMBL2199169 0.88 PLK1 (0.43) ALDH1A1HPGDSMN1; SMN2PLK1RPS6KB1
SCHEMBL2197926 0.88 PLK1 (0.37) ALDH1A1HPGDKDM4ESMN1; SMN2PLK1
SCHEMBL3559127 0.87 CDK2 (0.37) ALDH1A1HPGDPLK1RPS6KB1CDK1
SCHEMBL2200194 0.86 VNN1 (0.36) ALDH1A1HPGDKDM4ESMN1; SMN2PLK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2116543-A1 NOVEL AMINOPYRIMIDINE DERIVATIVE AS PLK1 INHIBITOR BANYU PHARMACEUTICAL CO., LTD. (JP) 2009-11-11 EP disclosed