SCHEMBL4258583

SCHEMBL4258583

O=C(NC(F)(F)F)c1ccc(F)cc1C(F)(F)F.O=S(=O)(O)/C=C/c1cccnc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NFE2L2 Q16236 3/20 0.45
ALDH1A1 P00352 1/20 0.43
NAMPT P43490 11/20 0.41
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
RAB9A P51151 1/20 0.38
HDAC3 O15379 1/20 0.38
NCOR1 O75376 1/20 0.38
HDAC4 P56524 1/20 0.38
KCNH2 Q12809 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC7 Q8WUI4 1/20 0.38
HDAC2 Q92769 1/20 0.38
HDAC10 Q969S8 1/20 0.38
HDAC11 Q96DB2 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
HDAC9 Q9UKV0 1/20 0.38
HDAC5 Q9UQL6 1/20 0.38
AURKA O14965 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27706035 0.87 NFE2L2 (0.47) NFE2L2ALDH1A1NAMPTMEN1KMT2A
SCHEMBL4263131 0.87 NFE2L2 (0.47) NFE2L2ALDH1A1NAMPTMEN1KMT2A
SCHEMBL4265094 0.85 NFE2L2 (0.47) NFE2L2ALDH1A1NAMPTMEN1KMT2A
SCHEMBL4265100 0.85 NFE2L2 (0.47) NFE2L2ALDH1A1NAMPTMEN1KMT2A
SCHEMBL4258585 0.77 NFE2L2 (0.46) NFE2L2ALDH1A1NAMPTMEN1KMT2A
SCHEMBL4261210 0.77 NAMPT (0.45) NFE2L2NAMPTHDAC3ALOX5PTGS1
SCHEMBL4262713 0.75 NFE2L2 (0.50) NFE2L2ALDH1A1NAMPTMEN1KMT2A
SCHEMBL27726712 0.75 NFE2L2 (0.50) NFE2L2ALDH1A1NAMPTMEN1KMT2A
SCHEMBL4262721 0.75 FLT1 (0.47) NFE2L2NAMPTHDAC3FLT4
SCHEMBL4620011 0.73 HTR2A (0.41) ALDH1A1MEN1KMT2AKCNH2PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1904471-B1 HETEROARYLETHENYL DERIVATIVES, THEIR MANUFACTURE AND USE AS PHARMACEUTICAL AGENTS HOFFMANN LA ROCHE (CH) 2009-10-21 EP disclosed