SCHEMBL4259674

SCHEMBL4259674

Fc1cnc(-c2ccc3[nH]ccc3c2)o1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APP P05067 2/20 0.56
PSMB8 P28062 1/20 0.52
NPC1 O15118 1/20 0.46
AHR P35869 1/20 0.46
LRRK2 Q5S007 4/20 0.46
S1PR1 P21453 2/20 0.44
MAP3K11 Q16584 2/20 0.44
BRD4 O60885 1/20 0.43
S1PR3 Q99500 1/20 0.43
GUSB P08236 1/20 0.43
FYN P06241 1/20 0.43
NISCH Q9Y2I1 1/20 0.42
CYP17A1 P05093 1/20 0.41
CYP11B1 P15538 1/20 0.41
CYP11B2 P19099 1/20 0.41
DYRK3 O43781 1/20 0.41
CCNT1 O60563 1/20 0.41
CCNA2 P20248 1/20 0.41
CDK2 P24941 1/20 0.41
CDK9 P50750 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7122837 0.72 PSMB8 (0.51) APPPSMB8NPC1AHRLRRK2
SCHEMBL30439233 0.72 PSMB8 (0.51) APPPSMB8NPC1AHRLRRK2
SCHEMBL5850255 0.72 NPC1 (0.79) PSMB8NPC1AHRMAP3K11BRD4
SCHEMBL1507829 0.71 APP (1.00) APPPSMB8NPC1AHR
SCHEMBL18284268 0.70 BRD4 (0.50) APPPSMB8AHRLRRK2S1PR1
SCHEMBL12615888 0.70 NOTUM (0.61) APPPSMB8
SCHEMBL856313 0.70 AHR (0.70) APPNPC1AHRMAP3K11GUSB
SCHEMBL10187349 0.69 MAP3K11 (0.52) NPC1AHRLRRK2MAP3K11BRD4
SCHEMBL12680497 0.68 NPC1 (0.56) NPC1AHRLRRK2MAP3K11FYN
SCHEMBL14365330 0.68 MAP3K11 (0.67) NPC1LRRK2MAP3K11FYNDYRK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009155017-A2 NOVEL SUBSTITUTED AZABENZOXAZOLES MERCK & CO., INC. (US) 2009-12-23 WO disclosed