SCHEMBL4263538

SCHEMBL4263538

CC(C)(CC(=O)OCC1c2ccccc2-c2ccccc21)OC(=O)CN

nearest known ligand 0.51

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.51
FABP5 Q01469 3/20 0.41
FABP7 O15540 2/20 0.41
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
EPHX2 P34913 1/20 0.40
HTR2A P28223 1/20 0.38
CASP3 P42574 1/20 0.36
MDM4 O15151 1/20 0.35
TP53 P04637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31047777 0.90 KMT2A (0.44) KMT2AFABP5FABP7CA1CA2
SCHEMBL28458423 0.90 KMT2A (0.44) KMT2AFABP5FABP7CA1CA2
SCHEMBL4690511 0.85 KMT2A (0.47) KMT2AFABP5FABP7CA1CA2
SCHEMBL12187737 0.83 KMT2A (0.64) KMT2AFABP5FABP7CA1CA2
SCHEMBL30935801 0.82 FABP5 (0.43) KMT2AFABP5FABP7CA1CA2
SCHEMBL31540857 0.82 KMT2A (0.50) KMT2AFABP5FABP7CA1CA2
Hydrochloric Acid SCHEMBL18981946 0.82 KMT2A (0.62) KMT2AFABP5FABP7CA1CA2
Hydrochloric Acid SCHEMBL31540856 0.81 KMT2A (0.49) KMT2AFABP5FABP7CA1CA2
SCHEMBL9511258 0.81 CASP3 (0.44) KMT2AFABP5FABP7CA1CA2
SCHEMBL26941528 0.81 KMT2A (0.48) KMT2AFABP5FABP7CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2114958-A1 INHIBITORS OF SERINE PROTEASES FOR THE TREATMENT OF HCV INFECTIONS Vertex Pharmceuticals Incorporated (US) 2009-11-11 EP disclosed
WO-2008106139-A1 INHIBITORS OF SERINE PROTEASES FOR THE TREATMENT OF HCV INFECTIONS VERTEX PHARMACEUTICALS INCORPORATED (US) 2008-09-04 WO disclosed