SCHEMBL9511258

SCHEMBL9511258

CC(C)(CC(=O)OCC1c2ccccc2-c2ccccc21)OC(=O)[C@@H](N)CC(=O)O

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 4/20 0.44
KMT2A Q03164 2/20 0.40
FABP5 Q01469 3/20 0.40
FABP7 O15540 2/20 0.40
CYP1A2 P05177 1/20 0.38
TSHR P16473 1/20 0.38
EPHX2 P34913 1/20 0.36
MDM4 O15151 1/20 0.36
TP53 P04637 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30983194 0.82 CASP3 (0.50) CASP3KMT2AFABP5FABP7CYP1A2
SCHEMBL9188706 0.82 CASP3 (0.50) CASP3KMT2AFABP5FABP7CYP1A2
SCHEMBL7123965 0.82 CASP3 (0.50) CASP3KMT2AFABP5FABP7CYP1A2
SCHEMBL4263538 0.81 KMT2A (0.51) CASP3KMT2AFABP5FABP7EPHX2
SCHEMBL28458423 0.81 KMT2A (0.44) CASP3KMT2AFABP5FABP7EPHX2
SCHEMBL31047777 0.81 KMT2A (0.44) CASP3KMT2AFABP5FABP7EPHX2
SCHEMBL4690511 0.79 KMT2A (0.47) CASP3KMT2AFABP5FABP7CYP1A2
SCHEMBL30935801 0.79 FABP5 (0.43) CASP3KMT2AFABP5FABP7EPHX2
SCHEMBL1096890 0.77 CASP3 (0.44) CASP3KMT2AEPHX2MDM4TP53
SCHEMBL31540857 0.77 KMT2A (0.50) CASP3KMT2AFABP5FABP7CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0401177-B1 SYNTHETIC PEPTIDE ANTAGONISTS OF NEUROKININ A, SALTS THEREOF AND RESPECTIVE PREPARATION PROCESSES A. MENARINI INDUSTRIE FARMACEUTICHE RIUNITE S.R.L. (IT) 1993-09-08 EP disclosed
US-5128447-A Bronchodilation, antispasmodic for intestines or bladder A. MENARINI INDUSTRIE FARMACEUTICHE RIUNITE S.R.L. (IT) 1992-07-07 US disclosed
EP-0401177-A1 Synthetic peptide antagonists of neurokinin A, salts thereof and respective preparation processes A. MENARINI INDUSTRIE FARMACEUTICHE RIUNITE S.R.L. (IT) 1990-12-05 EP disclosed