SCHEMBL4267443

SCHEMBL4267443

Cc1c(Cl)c2c3c(ccc2n1S(=O)(=O)c1cccc(F)c1)OCCNC3

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.42
PKLR P30613 1/20 0.42
HTR6 P50406 16/20 0.41
PTGDR Q13258 1/20 0.40
PTGDR2 Q9Y5Y4 1/20 0.40
HTT P42858 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
KMT2A Q03164 1/20 0.36
HTR1A P08908 1/20 0.35
DRD2 P14416 1/20 0.35
HTR7 P34969 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2003457 0.71 HTR6 (0.46) PKMPKLRHTR6
SCHEMBL1999781 0.69 HTR6 (0.46) PKMPKLRHTR6
SCHEMBL1997804 0.69 HTR6 (0.43) PKMPKLRHTR6
SCHEMBL2001693 0.68 HTR6 (0.46) PKMPKLRHTR6
Trifluoroacetic Acid SCHEMBL1993157 0.67 HTR6 (0.41) PKMPKLRHTR6PTGDRPTGDR2
SCHEMBL2001918 0.66 PKM (0.44) PKMPKLRHTR6HTTSMN1; SMN2
Trifluoroacetic Acid SCHEMBL2000044 0.65 HTR6 (0.39) PKMPKLRHTR6
Trifluoroacetic Acid SCHEMBL1998224 0.65 HTR6 (0.40) PKMPKLRHTR6
SCHEMBL1997377 0.65 HTR6 (0.40) HTR6
SCHEMBL1994607 0.65 HTR6 (0.42) HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2091953-A1 8-SULFONYL-L, 3, 4, 8-TETRAHYDR0-2H- [1, 4]OXAZEPINO [6, 7-E]INDOLE DERIVATIVES AND THEIR USE AS 5-HT6 RECEPTOR LIGANDS BIOVITRUM AB (publ) (SE) 2009-08-26 EP disclosed
WO-2008054288-A1 8-SULFONYL-L, 3, 4, 8-TETRAHYDR0-2H- [1, 4] OXAZEPINO [6, 7-E] INDOLE DERIVATIVES AND THEIR USE AS 5-HT6 RECEPTOR LIGANDS BIOVITRUM AB (PUBL) (SE) 2008-05-08 WO disclosed