Prifelone

Prifelone

SCHEMBL42678

CC(C)(C)c1cc(C(=O)c2cccs2)cc(C(C)(C)C)c1O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 4/20 1.00
PTGS2 P35354 4/20 1.00
ALOX5 P09917 3/20 1.00
HPGDS O60760 1/20 0.56
CNR2 P34972 7/20 0.52
CNR1 P21554 3/20 0.52
HPGD P15428 3/20 0.51
HTT P42858 1/20 0.51
CYP2C9 P11712 2/20 0.48
LMNA P02545 1/20 0.48
KDM4E B2RXH2 1/20 0.48
ALDH1A1 P00352 1/20 0.48
RXFP1 Q9HBX9 1/20 0.48
NPC1 O15118 1/20 0.48
TSHR P16473 1/20 0.48
RAB9A P51151 1/20 0.48
CA2 P00918 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Dimethylamine SCHEMBL10428349 0.89 ALOX5 (0.79) PTGS1PTGS2ALOX5HPGDSCNR2
Hydrochloric Acid SCHEMBL10428299 0.87 ALOX5 (0.75) PTGS1PTGS2ALOX5HPGDSCNR2
SCHEMBL10428667 0.86 PTGS1 (0.75) PTGS1PTGS2ALOX5HPGDSCNR2
SCHEMBL10428348 0.85 ALOX5 (0.73) PTGS1PTGS2ALOX5HPGDSCNR2
SCHEMBL10428259 0.85 ALOX5 (0.73) PTGS1PTGS2ALOX5HPGDSCNR2
Diethylamine SCHEMBL10428417 0.83 ALOX5 (0.70) PTGS1PTGS2ALOX5HPGDSCNR2
Hydrochloric Acid SCHEMBL10428718 0.83 PTGS1 (0.70) PTGS1PTGS2ALOX5HPGDSCNR2
Hydrochloric Acid SCHEMBL10428416 0.83 ALOX5 (0.68) PTGS1PTGS2ALOX5HPGDSCNR2
SCHEMBL10428256 0.82 ALOX5 (0.67) PTGS1PTGS2ALOX5HTTKDM4E
Hydrochloric Acid SCHEMBL10428717 0.82 PTGS1 (0.67) PTGS1PTGS2ALOX5HPGDSCNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2928 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118141602-A Lacrimal canaliculus embolism 上海曙瑞科技有限公司 2024-06-07 CN claimed
EP-4335413-A2 PROSTHETIC TISSUE VALVES Cormatrix Cardiovascular, Inc. (US) 2024-03-13 EP claimed
WO-2023212179-A2 THERAPEUTIC COMPOSITIONS FOR SKIN DISORDERS AND WOUND REPAIR UNIVERSITY OF MIAMI (US) 2023-11-02 WO claimed
CN-112575116-B Soybean whole genome SNP locus combination, gene chip and application 中国科学院东北地理与农业生态研究所 2023-05-12 CN claimed
US-20220110979-A1 FIBROBLAST REGENERATIVE CELLS FIGENE, LLC 2022-04-14 US claimed
EP-3908297-A1 FIBROBLAST REGENERATIVE CELLS Figene, LLC (US) 2021-11-17 EP claimed
EP-3279663-B1 USE OF GELSOLIN TO DIAGNOSE AND TREAT INFLAMMATORY DISEASES BRIGHAM & WOMENS HOSPITAL INC (US) 2021-07-28 EP claimed
WO-2020146874-A1 FIBROBLAST REGENERATIVE CELLS FIGENE, LLC (US) 2020-07-16 WO claimed
US-10377779-B2 Carbonate prodrugs and methods of using the same ACORDA THERAPEUTICS, INC. (US) 2019-08-13 US claimed
US-20180086778-A1 CARBONATE PRODRUGS AND METHODS OF USING THE SAME NEUROGESX, INC. 2018-03-29 US claimed
EP-1003501-A4 MEANS OF ASCERTAINING AN INDIVIDUAL'S RISK PROFILE FOR ATHEROSCLEROTIC DISEASE BRIGHAM & WOMENS HOSPITAL (US) 2001-01-17 EP claimed
EP-0707446-A4 PHARMACEUTICAL COMPOSITIONS AND USE THEREOF FOR TREATMENT OF NEUROLOGICAL DISEASES AND ETIOLOGICALLY RELATED SYMPTOMOLOGY SHAPIRO HOWARD K (US) 2001-01-10 EP claimed
EP-1003501-A1 MEANS OF ASCERTAINING AN INDIVIDUAL'S RISK PROFILE FOR ATHEROSCLEROTIC DISEASE BRIGHAM AND WOMEN'S HOSPITAL, INC. (US) 2000-05-31 EP claimed
WO-1998043630-A1 MEANS OF ASCERTAINING AN INDIVIDUAL'S RISK PROFILE FOR ATHEROSCLEROTIC DISEASE BRIGHAM AND WOMEN'S HOSPITAL, INC. (US) 1998-10-08 WO claimed
JP-H08512055-A 1996-12-17 JP claimed
EP-0707446-A1 PHARMACEUTICAL COMPOSITIONS AND USE THEREOF FOR TREATMENT OF NEUROLOGICAL DISEASES AND ETIOLOGICALLY RELATED SYMPTOMOLOGY SHAPIRO, Howard, K. (US) 1996-04-24 EP claimed
WO-1995001096-A1 PHARMACEUTICAL COMPOSITIONS AND USE THEREOF FOR TREATMENT OF NEUROLOGICAL DISEASES AND ETIOLOGICALLY RELATED SYMPTOMOLOGY SHAPIRO HOWARD K (US) 1995-01-12 WO claimed
US-4738842-A CONTAINING 2,6-DI-TERT-BUTYL-4-(2*-THENOYL) PHENOL RIKER LABORATORIES (US) 1988-04-19 US claimed
US-4212882-A ANTIINFLAMMATORY INTERMEDIATES RIKER LABORATORIES, INC. (US) 1980-07-15 US claimed
US-4172082-A ANTIINFLAMMATORY AGENTS RIKER LABORATORIES, INC. (US) 1979-10-23 US claimed