SCHEMBL4268356

SCHEMBL4268356

CC(=O)OOc1cc(CCCNCCC(c2ccccc2)c2ccccc2)ccc1F

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.50
MTNR1A P48039 3/20 0.40
MTNR1B P49286 3/20 0.40
SIGMAR1 Q99720 1/20 0.38
HDAC3 O15379 3/20 0.38
HDAC4 P56524 3/20 0.38
HDAC1 Q13547 3/20 0.38
HDAC7 Q8WUI4 3/20 0.38
HDAC2 Q92769 3/20 0.38
HDAC10 Q969S8 3/20 0.38
HDAC11 Q96DB2 3/20 0.38
HDAC8 Q9BY41 3/20 0.38
HDAC6 Q9UBN7 3/20 0.38
HDAC9 Q9UKV0 3/20 0.38
HDAC5 Q9UQL6 3/20 0.38
CYP4F2 P78329 1/20 0.38
CYP4A11 Q02928 1/20 0.38
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
CALM1 P0DP23 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4268359 0.89 KCNH2 (0.52) KCNH2MTNR1AMTNR1BSIGMAR1HDAC3
SCHEMBL3172754 0.83 KCNH2 (0.52) KCNH2SIGMAR1HDAC3HDAC4HDAC1
SCHEMBL4268708 0.82 KCNH2 (0.56) KCNH2MTNR1AMTNR1BSIGMAR1
SCHEMBL4275377 0.81 MTNR1A (0.35) MTNR1AMTNR1BCYP4F2CYP4A11MEN1
SCHEMBL4275384 0.80 PTGDR2 (0.55) MEN1KMT2A
SCHEMBL4266924 0.76 CYP4A11 (0.52) MTNR1AMTNR1BCYP4F2CYP4A11
SCHEMBL4268711 0.75 KCNH2 (0.59) KCNH2MTNR1AMTNR1BSIGMAR1
SCHEMBL4275709 0.75 CYP4F2 (0.48) MTNR1AMTNR1BCYP4F2CYP4A11
SCHEMBL16501807 0.70 KCNH2 (0.67) KCNH2SIGMAR1HDAC3HDAC4HDAC1
SCHEMBL4275379 0.69 PTGDR2 (0.56) CYP4F2CYP4A11MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2094662-A1 POLYCYCLIC ACID COMPOUNDS USEFUL AS CRTH2 ANTAGONISTS AND ANTIALLERGIC AGENTS Astellas Pharma Inc. (JP) 2009-09-02 EP disclosed
WO-2008072784-A1 POLYCYCLIC ACID COMPOUNDS USEFUL AS CRTH2 ANTAGONISTS AND ANTIALLERGIC AGENTS ASTELLAS PHARMA INC. (JP) 2008-06-19 WO disclosed