Cloticasone Propionate

Cloticasone Propionate

SCHEMBL42706

CCC(=O)O[C@]1(C(=O)SCCl)[C@H](C)C[C@H]2[C@@H]3C[C@H](F)C4=CC(=O)C=C[C@]4(C)[C@@]3(F)[C@@H](O)C[C@@]21C

nearest known ligand 0.87

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 13/20 0.87
PGR P06401 6/20 0.87
CYP3A4 P08684 6/20 0.87
AR P10275 5/20 0.87
ADORA3 P0DMS8 2/20 0.87
NR3C2 P08235 2/20 0.87
NR1I2 O75469 2/20 0.87
CHRM1 P11229 1/20 0.81
ADRA1A P35348 1/20 0.81
CNR1 P21554 1/20 0.66
PTGS1 P23219 1/20 0.66
HIF1A Q16665 3/20 0.64
SMN1; SMN2 Q16637 3/20 0.64
ALDH1A1 P00352 2/20 0.64
CYP1A2 P05177 1/20 0.64
LMNA P02545 2/20 0.61
USP2 O75604 2/20 0.61
ABCB11 O95342 2/20 0.61
MAPT P10636 2/20 0.61
MLNR O43193 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Cloticasone Propionate SCHEMBL15311037 1.00 NR3C1 (0.87) NR3C1PGRCYP3A4ARADORA3
Cloticasone Propionate SCHEMBL14518229 1.00 NR3C1 (0.87) NR3C1PGRCYP3A4ARADORA3
Cloticasone Propionate SCHEMBL13773292 1.00 NR3C1 (0.87) NR3C1PGRCYP3A4ARADORA3
Cloticasone Propionate SCHEMBL1860078 1.00 NR3C1 (0.87) NR3C1PGRCYP3A4ARADORA3
Cloticasone Propionate SCHEMBL15311035 1.00 NR3C1 (0.87) NR3C1PGRCYP3A4ARADORA3
Cloticasone Propionate SCHEMBL17735459 1.00 NR3C1 (0.87) NR3C1PGRCYP3A4ARADORA3
SCHEMBL14479087 0.94 NR3C1 (0.90) NR3C1PGRCYP3A4ARADORA3
SCHEMBL195423 0.94 NR3C1 (0.90) NR3C1PGRCYP3A4ARADORA3
Fluticasone Propionate SCHEMBL14339613 0.93 NR3C1 (1.00) NR3C1PGRCYP3A4ARADORA3
Fluticasone Propionate SCHEMBL5482829 0.93 NR3C1 (1.00) NR3C1PGRCYP3A4ARADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2676 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4335413-A2 PROSTHETIC TISSUE VALVES Cormatrix Cardiovascular, Inc. (US) 2024-03-13 EP claimed
WO-2023212179-A2 THERAPEUTIC COMPOSITIONS FOR SKIN DISORDERS AND WOUND REPAIR UNIVERSITY OF MIAMI (US) 2023-11-02 WO claimed
US-20220110979-A1 FIBROBLAST REGENERATIVE CELLS FIGENE, LLC 2022-04-14 US claimed
EP-3908297-A1 FIBROBLAST REGENERATIVE CELLS Figene, LLC (US) 2021-11-17 EP claimed
EP-3279663-B1 USE OF GELSOLIN TO DIAGNOSE AND TREAT INFLAMMATORY DISEASES BRIGHAM & WOMENS HOSPITAL INC (US) 2021-07-28 EP claimed
WO-2020146874-A1 FIBROBLAST REGENERATIVE CELLS FIGENE, LLC (US) 2020-07-16 WO claimed
EP-3279663-A1 USE OF GELSOLIN TO DIAGNOSE AND TREAT INFLAMMATORY DISEASES The Brigham and Women's Hospital, Inc. (US) 2018-02-07 EP claimed
US-20170281724-A9 USE OF GELSOLIN TO DIAGNOSE AND TREAT INFLAMMATORY DISEASES THE BRIGHAM AND WOMEN'S HOSPITAL, INC. (US) 2017-10-05 US claimed
EP-2001496-B1 USE OF GELSOLIN TO DIAGNOSE AND TREAT INFLAMMATORY DISEASES BRIGHAM & WOMENS HOSPITAL INC (US) 2017-05-31 EP claimed
US-20160228505-A1 USE OF GELSOLIN TO DIAGNOSE AND TREAT INFLAMMATORY DISEASES THE BRIGHAM AND WOMEN'S HOSPITAL, INC. (US) 2016-08-11 US claimed
WO-2003088811-A2 GELSOLIN AS A PROGNOSTIC MARKER OF ARTHEROSCLEROTIC DISEASES THE BRIGHAM AND WOMEN'S HOSPITAL, INC. (US) 2003-10-30 WO claimed
US-20030152566-A1 Soluble CD40L (CD154) as a prognostic marker of atherosclerotic diseases THE BRIGHAM AND WOMEN'S HOSPITAL, INC. (US) 2003-08-14 US claimed
WO-2003040691-A2 SOLUBLE CD40L(CD154) AS A PROGNOSTIC MARKER OF ATHEROSCLEROTIC DISEASES THE BRIGHAM AND WOMEN'S HOSPITAL, INC. (US) 2003-05-15 WO claimed
WO-2001015744-A9 SYSTEMIC INFLAMMATORY MARKERS AS DIAGNOSTIC TOOLS IN THE PREVENTION OF ATHEROSCLEROTIC DISEASES BRIGHAM & WOMENS HOSPITAL (US) 2002-09-26 WO claimed
EP-1212101-A1 SYSTEMIC INFLAMMATORY MARKERS AS DIAGNOSTIC TOOLS IN THE PREVENTION OF ATHEROSCLEROTIC DISEASES THE BRIGHAM AND WOMEN'S HOSPITAL, INC. (US) 2002-06-12 EP claimed
JP-2001525058-A 2001-12-04 JP claimed
WO-2001015744-A1 SYSTEMIC INFLAMMATORY MARKERS AS DIAGNOSTIC TOOLS IN THE PREVENTION OF ATHEROSCLEROTIC DISEASES THE BRIGHAM AND WOMEN'S HOSPITAL, INC. (US) 2001-03-08 WO claimed
EP-1003501-A4 MEANS OF ASCERTAINING AN INDIVIDUAL'S RISK PROFILE FOR ATHEROSCLEROTIC DISEASE BRIGHAM & WOMENS HOSPITAL (US) 2001-01-17 EP claimed
EP-1003501-A1 MEANS OF ASCERTAINING AN INDIVIDUAL'S RISK PROFILE FOR ATHEROSCLEROTIC DISEASE BRIGHAM AND WOMEN'S HOSPITAL, INC. (US) 2000-05-31 EP claimed
WO-1998043630-A1 MEANS OF ASCERTAINING AN INDIVIDUAL'S RISK PROFILE FOR ATHEROSCLEROTIC DISEASE BRIGHAM AND WOMEN'S HOSPITAL, INC. (US) 1998-10-08 WO claimed