SCHEMBL4275871

SCHEMBL4275871

COc1ccccc1Cc1sc(NC(=O)c2ccc3c(c2)CCNC3)nc1C

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 5/20 0.46
ROCK2 O75116 3/20 0.46
SMN1; SMN2 Q16637 6/20 0.45
MAPT P10636 2/20 0.45
RAB9A P51151 2/20 0.45
NPC1 O15118 1/20 0.45
LMNA P02545 2/20 0.44
KMT2A Q03164 2/20 0.44
MEN1 O00255 1/20 0.44
PRKG1 Q13976 1/20 0.42
ALDH1A1 P00352 4/20 0.41
TP53 P04637 1/20 0.41
KDM4E B2RXH2 4/20 0.41
HTT P42858 2/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
ROCK1 Q13464 1/20 0.41
CYP3A4 P08684 1/20 0.41
PTGER1 P34995 2/20 0.40
HTR2C P28335 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4278219 0.99 HPGD (0.46) HPGDROCK2SMN1; SMN2MAPTRAB9A
SCHEMBL13573324 0.90 HPGD (0.45) HPGDROCK2SMN1; SMN2MAPTRAB9A
SCHEMBL4282701 0.90 PTGER1 (0.53) HPGDROCK2SMN1; SMN2MAPTRAB9A
Hydrochloric Acid SCHEMBL4283252 0.89 PTGER1 (0.54) HPGDROCK2SMN1; SMN2MAPTRAB9A
SCHEMBL4285373 0.87 SMN1; SMN2 (0.45) HPGDROCK2SMN1; SMN2MAPTRAB9A
Hydrochloric Acid SCHEMBL4279458 0.86 SMN1; SMN2 (0.44) HPGDROCK2SMN1; SMN2MAPTRAB9A
SCHEMBL4282184 0.86 HPGD (0.52) HPGDROCK2SMN1; SMN2MAPTRAB9A
Hydrochloric Acid SCHEMBL4287316 0.85 HPGD (0.52) HPGDROCK2SMN1; SMN2MAPTRAB9A
SCHEMBL4274873 0.84 SMN1; SMN2 (0.48) HPGDROCK2SMN1; SMN2MAPTRAB9A
Hydrochloric Acid SCHEMBL4279972 0.84 SMN1; SMN2 (0.47) HPGDROCK2SMN1; SMN2MAPTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009150196-A1 N-THIAZOLYL-1, 2, 3, 4-TETRAHYDRO-6-ISOQUINOLINECARBOXAMIDE DERIVATIVES AS INHIBITORS OF STEAROYL COENZYME A DESATURASE SMITHKLINE BEECHAM CORPORATION (US) 2009-12-17 WO claimed
WO-2009150196-A1 N-THIAZOLYL-1, 2, 3, 4-TETRAHYDRO-6-ISOQUINOLINECARBOXAMIDE DERIVATIVES AS INHIBITORS OF STEAROYL COENZYME A DESATURASE SMITHKLINE BEECHAM CORPORATION (US) 2009-12-17 WO disclosed