SCHEMBL4278175

SCHEMBL4278175

COc1cc2c(cc1OC)CCC(C=CC(=O)N(C(C)C)C(C)C)=C2

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.37
MEN1 O00255 3/20 0.36
KMT2A Q03164 3/20 0.36
PTGS2 P35354 2/20 0.36
APP P05067 1/20 0.35
LMNA P02545 1/20 0.35
PTGS1 P23219 2/20 0.34
ATM Q13315 1/20 0.34
HPGD P15428 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
MAOA P21397 3/20 0.33
KDM4E B2RXH2 2/20 0.33
GLA P06280 2/20 0.33
ACHE P22303 2/20 0.33
MAOB P27338 2/20 0.33
GABRA1 P14867 1/20 0.33
GABRB2 P47870 1/20 0.33
BCHE P06276 1/20 0.32
PTGES O14684 1/20 0.32
ALOX5 P09917 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4278171 1.00 ALDH1A1 (0.37) ALDH1A1MEN1KMT2APTGS2APP
SCHEMBL4427869 0.82 ALDH1A1 (0.36) ALDH1A1KMT2APTGS2LMNAHPGD
SCHEMBL4269322 0.82 KDM4E (0.47) ALDH1A1MEN1KMT2APTGS2LMNA
SCHEMBL4269325 0.82 KDM4E (0.47) ALDH1A1MEN1KMT2APTGS2LMNA
SCHEMBL4279861 0.81 RECQL (0.47) ALDH1A1MEN1KMT2APTGS2LMNA
SCHEMBL4279859 0.81 RECQL (0.47) ALDH1A1MEN1KMT2APTGS2LMNA
SCHEMBL4266223 0.80 TRPV1 (0.51) ALDH1A1KMT2APTGS2LMNAHPGD
SCHEMBL4266221 0.80 TRPV1 (0.51) ALDH1A1KMT2APTGS2LMNAHPGD
Pyrrole SCHEMBL4270409 0.77 ALDH1A1 (0.40) ALDH1A1MEN1KMT2APTGS2LMNA
SCHEMBL4266849 0.77 TRPM8 (0.36) MEN1KMT2APTGS2LMNAPTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009110002-A1 NOVEL EFFLUX PUMP INHIBITORS COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2009-09-11 WO claimed