SCHEMBL4279472

SCHEMBL4279472

N/C(=N\O)c1ccc2c(c1)CCN2

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.51
DRD4 P21917 1/20 0.51
KDM4E B2RXH2 1/20 0.47
MAPT P10636 1/20 0.47
ALDH1A1 P00352 1/20 0.40
CYP2C9 P11712 1/20 0.40
ALOX15 P16050 1/20 0.40
CYP2C19 P33261 1/20 0.40
CRBN Q96SW2 1/20 0.38
RECQL P46063 1/20 0.38
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA9 Q16790 1/20 0.36
PLAU P00749 1/20 0.36
NNMT P40261 1/20 0.36
ACHE P22303 4/20 0.36
KDM1A O60341 1/20 0.35
SIRT2 Q8IXJ6 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4279479 1.00 DRD2 (0.51) DRD2DRD4KDM4EMAPTALDH1A1
SCHEMBL4051485 0.79 KDM4E (0.58) DRD2DRD4KDM4EMAPTALDH1A1
SCHEMBL29673233 0.79 DRD2 (0.55) DRD2DRD4KDM4EMAPTALDH1A1
SCHEMBL18175179 0.79 DRD2 (0.55) DRD2DRD4KDM4EMAPTALDH1A1
SCHEMBL29779540 0.79 KDM4E (0.58) DRD2DRD4KDM4EMAPTALDH1A1
Hydrochloric Acid SCHEMBL30263125 0.78 KDM4E (0.57) DRD2DRD4KDM4EMAPTALDH1A1
SCHEMBL773530 0.75 PNMT (0.49) DRD2
SCHEMBL773531 0.75 PNMT (0.49) DRD2
SCHEMBL772706 0.75 PLAU (0.49) DRD2PLAU
SCHEMBL772707 0.75 PLAU (0.49) DRD2PLAU

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009151621-A1 SUBSTITUTED (1, 2, 4-0XADIAZ0L-3-YL) INDOLIN-1-YL CARBOXYLIC ACID DERIVATIVES USEFUL AS S1P1 AGONISTS ARENA PHARMACEUTICALS, INC. (US) 2009-12-17 WO disclosed