SCHEMBL4281323

SCHEMBL4281323

O=C(Nc1ncc(Cc2ccc(Cl)c(Cl)c2)s1)c1ccc2c(c1)CCNC2

nearest known ligand 0.56

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SCD O00767 4/20 0.56
GAA P10253 1/20 0.47
SMN1; SMN2 Q16637 3/20 0.47
HSP90AA1 P07900 1/20 0.47
MAPT P10636 4/20 0.46
KMT2A Q03164 2/20 0.46
CYP1A2 P05177 2/20 0.46
LMNA P02545 2/20 0.46
MEN1 O00255 1/20 0.46
STAT3 P40763 1/20 0.44
CYP3A4 P08684 2/20 0.44
CYP2C19 P33261 1/20 0.44
HTT P42858 1/20 0.44
TP53 P04637 1/20 0.43
OGA O60502 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4289761 0.99 SCD (0.56) SCDGAASMN1; SMN2HSP90AA1MAPT
SCHEMBL4284053 0.91 GAA (0.57) SCDGAASMN1; SMN2MAPTKMT2A
Hydrochloric Acid SCHEMBL4276562 0.90 GAA (0.56) SCDGAASMN1; SMN2MAPTKMT2A
SCHEMBL4288598 0.88 KMT2A (0.61) SCDGAASMN1; SMN2MAPTKMT2A
Hydrochloric Acid SCHEMBL4279918 0.88 KMT2A (0.60) SCDGAASMN1; SMN2MAPTKMT2A
SCHEMBL4283271 0.87 POLB (0.56) SCDGAASMN1; SMN2MAPTKMT2A
SCHEMBL4284162 0.86 MAPT (0.61) SCDGAASMN1; SMN2MAPTKMT2A
Hydrochloric Acid SCHEMBL4279963 0.86 MAPT (0.60) SCDGAASMN1; SMN2MAPTKMT2A
SCHEMBL4277749 0.85 OGA (0.48) SCDGAASMN1; SMN2MAPTKMT2A
SCHEMBL4285057 0.85 MAPT (0.60) SCDGAASMN1; SMN2MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009150196-A1 N-THIAZOLYL-1, 2, 3, 4-TETRAHYDRO-6-ISOQUINOLINECARBOXAMIDE DERIVATIVES AS INHIBITORS OF STEAROYL COENZYME A DESATURASE SMITHKLINE BEECHAM CORPORATION (US) 2009-12-17 WO claimed
WO-2009150196-A1 N-THIAZOLYL-1, 2, 3, 4-TETRAHYDRO-6-ISOQUINOLINECARBOXAMIDE DERIVATIVES AS INHIBITORS OF STEAROYL COENZYME A DESATURASE SMITHKLINE BEECHAM CORPORATION (US) 2009-12-17 WO disclosed