SCHEMBL4282837

SCHEMBL4282837

CCCc1cc(N(CCCc2ccccc2)Cc2cccc(N3CCOCC3)c2)n(C)n1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 4/20 0.40
AGXT P21549 1/20 0.38
ALDH1A1 P00352 3/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
SIGMAR1 Q99720 4/20 0.37
POLB P06746 1/20 0.37
MAPT P10636 3/20 0.37
KDM4E B2RXH2 2/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
OPRM1 P35372 1/20 0.36
LMNA P02545 2/20 0.36
GAA P10253 1/20 0.36
HRH3 Q9Y5N1 1/20 0.35
NAPEPLD Q6IQ20 2/20 0.35
SLC16A3 O15427 1/20 0.35
SLC16A1 P53985 1/20 0.35
MCTS1 Q9ULC4 1/20 0.35
USP2 O75604 1/20 0.35
HPGD P15428 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4287197 0.82 AGXT (0.37) AGXTALDH1A1SMN1; SMN2MEN1KMT2A
SCHEMBL5141171 0.73 AGXT (0.40) AGXTMEN1KMT2ALMNASLC16A3
SCHEMBL8189516 0.70 AGXT (0.61) AGXTALDH1A1SMN1; SMN2SIGMAR1MAPT
SCHEMBL5141914 0.70 AGXT (0.39) AGXTMEN1KMT2ASLC16A3SLC16A1
SCHEMBL4507051 0.65 AGXT (0.65) AGXTALDH1A1SMN1; SMN2SIGMAR1MAPT
SCHEMBL5134153 0.64 GAA (0.41) ALDH1A1SMN1; SMN2POLBMAPTKDM4E
SCHEMBL17276273 0.63 AGXT (0.49) AGXTALDH1A1SMN1; SMN2MEN1KMT2A
SCHEMBL28276177 0.63 LMNA (0.55) AGXTALDH1A1SMN1; SMN2SIGMAR1MAPT
SCHEMBL26616472 0.63 POLB (0.50) ALDH1A1SMN1; SMN2SIGMAR1POLBMAPT
SCHEMBL18295011 0.63 AGXT (0.65) AGXTALDH1A1SIGMAR1MAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009071706-A1 PYRAZOLEPYRIMIDINE COMPOUNDS USEFUL FOR THE TREATMENT OF DEGENERATIVE & INFLAMMATORY DISEASES GALAPAGOS NV (BE) 2009-06-11 WO disclosed