Ethyl Biscoumacetate

Ethyl Biscoumacetate

SCHEMBL42830

CCOC(=O)C(c1c(O)c2ccccc2oc1=O)c1c(O)c2ccccc2oc1=O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 1/20 1.00
NQO1 P15559 4/20 0.76
ALDH1A1 P00352 2/20 0.64
CYP2C9 P11712 2/20 0.61
VKORC1 Q9BQB6 3/20 0.57
KDM4E B2RXH2 1/20 0.57
ALB P02768 1/20 0.57
PCSK7 Q16549 1/20 0.57
HSD17B10 Q99714 1/20 0.57
MEN1 O00255 1/20 0.57
KMT2A Q03164 1/20 0.57
TOP1 P11387 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ethyl Biscoumacetate SCHEMBL29359768 1.00 ADORA3 (1.00) ADORA3NQO1ALDH1A1CYP2C9VKORC1
SCHEMBL5107024 0.92 ADORA3 (0.86) ADORA3NQO1ALDH1A1CYP2C9VKORC1
Ethyl Biscoumacetate SCHEMBL1900704 0.87 ADORA3 (0.76) ADORA3NQO1ALDH1A1CYP2C9VKORC1
SCHEMBL1647635 0.87 ADORA3 (0.77) ADORA3NQO1ALDH1A1CYP2C9VKORC1
SCHEMBL14078678 0.83 ADORA3 (0.70) ADORA3NQO1ALDH1A1CYP2C9VKORC1
SCHEMBL5106117 0.83 ADORA3 (0.70) ADORA3NQO1ALDH1A1CYP2C9VKORC1
SCHEMBL1648320 0.82 ADORA3 (0.70) ADORA3NQO1ALDH1A1CYP2C9VKORC1
SCHEMBL14172135 0.81 NQO1 (0.72) ADORA3NQO1ALDH1A1CYP2C9VKORC1
SCHEMBL1647638 0.81 CYP2C9 (0.72) ADORA3NQO1ALDH1A1CYP2C9VKORC1
SCHEMBL1650108 0.81 ADORA3 (0.68) ADORA3NQO1ALDH1A1CYP2C9VKORC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2708 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250333462-A1 PERIOSTIN COMPOUNDS FOR THE TREATMENT OF HAEMATOLOGICAL COMPLICATIONS CHEMOTHERAPEUTISCHES FORSCHUNGSINSTITUT GEORG-SPEYER-HAUS (DE) 2025-10-30 US claimed
EP-3823660-B1 PERIOSTIN COMPOUNDS FOR THE TREATMENT OF HAEMATOLOGICAL COMPLICATIONS UNIV DER JOHANNES GUTENBERG UNIV MAINZ (DE) 2025-05-07 EP claimed
US-20240315965-A1 COMPOSITIONS AND METHODS RELATED TO PHARMACEUTICAL EXCIPIENTS Natural Extraction Systems, LLC (US) 2024-09-26 US claimed
US-11897969-B2 Inhibition of oxidation-specific epitopes to treat ischemic reperfusion injury THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2024-02-13 US claimed
US-20240034752-A1 ARTIFICIAL SHORT INTERFERING PEPTIDE FOR THE PHOSPHORYLATION SUBSTRATE OF DAPK1 AND ITS PHARMACEUTICAL APPLICATIONS BEIJING SINANCHENG TECHNOLOGY CO., LTD. (CN) 2024-02-01 US claimed
EP-4293037-A1 ARTIFICIAL SMALL MOLECULE INTERFERING PEPTIDE OF DAPK1 PHOSPHORYLATED SUBSTRATE AND PHARMACEUTICAL USE THEREOF Beijing Sinancheng Technology co., Ltd. (CN) 2023-12-20 EP claimed
US-20230089351-A1 METHODS RELATED TO BIOACTIVE AGENTS THAT CONVERT FROM ANIONS TO MOLECULES Natural Extraction Systems, LLC (US) 2023-03-23 US claimed
WO-2022182523-A1 COMPOSITIONS RELATED TO BIOACTIVE AGENTS THAT CONVERT FROM ANIONS TO MOLECULES Natural Extraction Systems, LLC (US) 2022-09-01 WO claimed
WO-2022182527-A1 COMPOSITIONS AND METHODS RELATED TO PHARMACEUTICAL EXCIPIENTS Natural Extraction Systems, LLC (US) 2022-09-01 WO claimed
US-11421234-B2 Aptamers for targeting coagulation factor XIII and uses thereof CHANG GUNG UNIVERSITY (TW) 2022-08-23 US claimed
EP-1218002-A1 USE OF FLAVONE 8-ACETIC ACID IN VASCULAR AND CARDIOVASCULAR INTERVENTIONS AND ACUTE CORONARY SYNDROMES Mruk, Jozef S. (US) 2002-07-03 EP claimed
EP-0951283-A4 NOVEL ARACHIDONIC ACID METABOLITE, 16-HETE UNIV VERMONT (US) 2002-06-26 EP claimed
US-20020071822-A1 Therapeutic polyesters and polyamides POLYMERIX CORPORATION 2002-06-13 US claimed
WO-2002009768-A2 THERAPEUTIC POLYESTERS AND POLYAMIDES RUTGERS, THE STATE UNIVERSITY (US) 2002-02-07 WO claimed
US-20010041687-A1 Use of flavone 8-acetic acid in vascular and cardiovascular interventions and acute coronary syndromes MRUK JOZEF S (US) 2001-11-15 US claimed
WO-2001052839-A1 USE OF FLAVONE 8-ACETIC ACID IN VASCULAR AND CARDIOVASCULAR INTERVENTIONS AND ACUTE CORONARY SYNDROMES MRUK JOZEF S (US) 2001-07-26 WO claimed
EP-0951283-A1 NOVEL ARACHIDONIC ACID METABOLITE, 16-HETE THE UNIVERSITY OF VERMONT (US) 1999-10-27 EP claimed
US-5753702-A INHIBITORS OF NEUTROPHIL ADHESION, ANTIINFLAMMATORY UNIVERSITY OF VERMONT (US) 1998-05-19 US claimed
WO-1997044024-A1 NOVEL ARACHIDONIC ACID METABOLITE, 16-HETE UNIVERSITY OF VERMONT (US) 1997-11-27 WO claimed
US-5130135-A Pyrethroids as insecticides SMITHKLINE BEECHAM PLC (GB) 1992-07-14 US claimed