SCHEMBL4283173

SCHEMBL4283173

Nc1ccc(Oc2ncnc3cc(CNC(=O)O)[nH]c23)cc1Cl

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KDR P35968 16/20 0.39
KIT P10721 2/20 0.39
PDGFRA P16234 2/20 0.39
FLT1 P17948 2/20 0.39
FLT4 P35916 2/20 0.39
CSF1R P07333 2/20 0.38
RET P07949 1/20 0.38
FLT3 P36888 1/20 0.38
KDM5A P29375 1/20 0.35
KDM4C Q9H3R0 1/20 0.35
KDM5B Q9UGL1 1/20 0.35
EGFR P00533 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4771434 0.81 EGFR (0.37) KDRKITPDGFRAFLT1FLT4
SCHEMBL4766245 0.80 KDM4C (0.34) KDRKITPDGFRAFLT1FLT4
SCHEMBL4282301 0.78 EGFR (0.41) KDRRETEGFR
SCHEMBL4290591 0.73 DYRK1A (0.45) KDREGFR
SCHEMBL4282048 0.73 KDR (0.49) KDREGFR
SCHEMBL4284118 0.73 RET (0.38) KDRKITPDGFRAFLT1FLT4
SCHEMBL4771430 0.71 EGFR (0.37) KDRKITPDGFRAFLT1FLT4
Hydrochloric Acid SCHEMBL4284171 0.67 KDR (0.65) KDRKITPDGFRAFLT1FLT4
SCHEMBL15960748 0.67 KDR (0.53) KDRKITPDGFRAFLT1FLT4
SCHEMBL4279915 0.66 KDR (0.46) KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090137580-A1 Fused Heterocyclic Derivatives and Use Thereof TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-05-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090137580-A1 Fused Heterocyclic Derivatives and Use Thereof TIE1, KDR, FLT1 KDR 2/4885KIT 30/4885PDGFRA 7/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.