SCHEMBL4283514

SCHEMBL4283514

O=C(Nc1csc(Cc2cccc(C(F)(F)F)c2)n1)c1ccc2c(c1)CCNC2

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
WNT1 P04628 2/20 0.44
GSK3B P49841 2/20 0.44
DYRK1A Q13627 2/20 0.44
CLK2 P49760 1/20 0.44
CLK3 P49761 1/20 0.44
ASIC3 Q9UHC3 1/20 0.43
SCD O00767 6/20 0.42
HTR2C P28335 2/20 0.42
HTR2B P41595 2/20 0.42
ROCK2 O75116 1/20 0.40
MAP3K5 Q99683 1/20 0.40
F2 P00734 1/20 0.40
PLG P00747 1/20 0.40
PLAU P00749 1/20 0.40
PLAT P00750 1/20 0.40
KLKB1 P03952 1/20 0.40
PRSS1 P07477 1/20 0.40
GPR52 Q9Y2T5 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4275852 0.99 WNT1 (0.44) WNT1GSK3BDYRK1ACLK2CLK3
SCHEMBL3729733 0.84 SCD (0.57) ASIC3SCDHTR2CHTR2B
Hydrochloric Acid SCHEMBL3725765 0.83 SCD (0.57) ASIC3SCDHTR2CHTR2B
SCHEMBL4288574 0.80 SCD (0.48) ASIC3SCDHTR2CHTR2BROCK2
SCHEMBL4275101 0.80 SCD (0.64) SCD
SCHEMBL13573288 0.80 ESR2 (0.43) SCDMAP3K5
Hydrochloric Acid SCHEMBL4275856 0.79 SCD (0.47) ASIC3SCDGPR52
Hydrochloric Acid SCHEMBL4276243 0.79 SCD (0.63) SCD
SCHEMBL20367363 0.78 WNT1 (0.44) WNT1GSK3BDYRK1ACLK2CLK3
SCHEMBL20162177 0.78 KDM4C (0.46) WNT1GSK3BDYRK1ACLK2CLK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009150196-A1 N-THIAZOLYL-1, 2, 3, 4-TETRAHYDRO-6-ISOQUINOLINECARBOXAMIDE DERIVATIVES AS INHIBITORS OF STEAROYL COENZYME A DESATURASE SMITHKLINE BEECHAM CORPORATION (US) 2009-12-17 WO claimed
WO-2009150196-A1 N-THIAZOLYL-1, 2, 3, 4-TETRAHYDRO-6-ISOQUINOLINECARBOXAMIDE DERIVATIVES AS INHIBITORS OF STEAROYL COENZYME A DESATURASE SMITHKLINE BEECHAM CORPORATION (US) 2009-12-17 WO disclosed
WO-2009150196-A1 N-THIAZOLYL-1, 2, 3, 4-TETRAHYDRO-6-ISOQUINOLINECARBOXAMIDE DERIVATIVES AS INHIBITORS OF STEAROYL COENZYME A DESATURASE SMITHKLINE BEECHAM CORPORATION (US) 2009-12-17 WO disclosed