SCHEMBL4288574

SCHEMBL4288574

Cc1sc(NC(=O)c2ccc3c(c2)CCNC3)nc1Cc1cccc(C(F)(F)F)c1

nearest known ligand 0.49

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SCD O00767 15/20 0.48
ASIC3 Q9UHC3 1/20 0.42
BTK Q06187 1/20 0.41
ROCK2 O75116 1/20 0.41
HTR2C P28335 1/20 0.41
HTR2B P41595 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4275856 0.88 SCD (0.47) SCDASIC3
SCHEMBL3729733 0.84 SCD (0.57) SCDASIC3HTR2CHTR2B
SCHEMBL4275101 0.83 SCD (0.64) SCD
Hydrochloric Acid SCHEMBL3725765 0.83 SCD (0.57) SCDASIC3HTR2CHTR2B
SCHEMBL4289707 0.83 PTGER1 (0.46) ROCK2
Hydrochloric Acid SCHEMBL4276243 0.83 SCD (0.63) SCD
Hydrochloric Acid SCHEMBL4279816 0.82 PTGER1 (0.46) ROCK2
SCHEMBL4283514 0.80 WNT1 (0.44) SCDASIC3ROCK2HTR2CHTR2B
Hydrochloric Acid SCHEMBL4275852 0.79 WNT1 (0.44) SCDASIC3ROCK2HTR2CHTR2B
SCHEMBL4283504 0.79 HPGD (0.47)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009150196-A1 N-THIAZOLYL-1, 2, 3, 4-TETRAHYDRO-6-ISOQUINOLINECARBOXAMIDE DERIVATIVES AS INHIBITORS OF STEAROYL COENZYME A DESATURASE SMITHKLINE BEECHAM CORPORATION (US) 2009-12-17 WO disclosed