Quinazoline

Quinazoline

SCHEMBL4283584

Oc1ccccc1O.c1ccc2ncncc2c1

nearest known ligand 0.80

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 10/20 0.80
PIK3CA P42336 2/20 0.53
PIK3CD O00329 1/20 0.53
KDM4E B2RXH2 3/20 0.41
MAPKAPK2 P49137 1/20 0.41
ALDH1A1 P00352 4/20 0.41
RAB9A P51151 3/20 0.41
NPC1 O15118 2/20 0.41
LMNA P02545 2/20 0.41
HPGD P15428 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
HTT P42858 1/20 0.41
GFER P55789 1/20 0.41
MAPT P10636 2/20 0.40
CA12 O43570 1/20 0.40
GMNN O75496 1/20 0.40
CA2 P00918 1/20 0.40
FYN P06241 1/20 0.40
POLB P06746 1/20 0.40
CA3 P07451 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Quinazoline SCHEMBL22833783 0.89 EGFR (1.00) EGFRPIK3CAPIK3CDKDM4EALDH1A1
Quinazoline SCHEMBL29356169 0.89 EGFR (1.00) EGFRPIK3CAPIK3CDKDM4EALDH1A1
Quinazoline SCHEMBL5920 0.89 EGFR (1.00) EGFRPIK3CAPIK3CDKDM4EALDH1A1
Quinazoline SCHEMBL29490398 0.89 EGFR (1.00) EGFRPIK3CAPIK3CDKDM4EALDH1A1
Quinazoline SCHEMBL561027 0.88 EGFR (0.67) EGFRPIK3CAPIK3CDKDM4EMAPKAPK2
Quinazoline SCHEMBL27275460 0.88 EGFR (0.87) EGFRPIK3CAPIK3CDALDH1A1CYP1A2
SCHEMBL3196932 0.87 EGFR (0.95) EGFRPIK3CAPIK3CDKDM4EALDH1A1
Quinazoline SCHEMBL3533306 0.87 EGFR (0.95) EGFRPIK3CAPIK3CDKDM4EALDH1A1
Quinazoline SCHEMBL4487630 0.87 EGFR (0.95) EGFRPIK3CAPIK3CDKDM4EALDH1A1
Quinazoline SCHEMBL21055790 0.87 EGFR (0.95) EGFRPIK3CAPIK3CDKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1797087-A4 CARBO- AND HETERO-CYCLIC ANTIBIOTICS AND USE THEREOF ULYSSES PHARMACEUTICAL PRODUCT (CA) 2009-06-03 EP disclosed
US-20080188499-A1 Carbo- and Hetero-Cyclic Antibiotics and Use Thereof ULYSSES PHARMACEUTICAL PRODUCTS INC. (CA) 2008-08-07 US disclosed
CN-101027299-A Carbon-and hetero-cyclic nitrofuran antibiotics and use thereof ULYSSES PHARMACEUTICAL PRODUCT (CA) 2007-08-29 CN disclosed
EP-1797087-A1 CARBO- AND HETERO-CYCLIC ANTIBIOTICS AND USE THEREOF Ulysses Pharmaceuticals Products Inc. (CA) 2007-06-20 EP disclosed
WO-2006032138-A1 CARBO- AND HETERO-CYCLIC ANTIBIOTICS AND USE THEREOF ULYSSES PHARMACEUTICAL PRODUCTS INC. (CA) 2006-03-30 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080188499-A1 Carbo- and Hetero-Cyclic Antibiotics and Use Thereof SLC7A1, CYP2C19, ABCB11 EGFR 720/4885PIK3CA 1343/4885PIK3CD 1074/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.