SCHEMBL4283690

SCHEMBL4283690

CCCC1CCCC(NC(=O)C(c2ccc(CN3N=C(c4ccccc4)OCC3=O)cc2)C(C)C)C1

nearest known ligand 0.35

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 3/20 0.35
ALDH1A1 P00352 2/20 0.34
HPGD P15428 2/20 0.34
TSHR P16473 2/20 0.34
ACKR3 P25106 1/20 0.34
CTSD P07339 2/20 0.32
MCHR1 Q99705 1/20 0.32
NR3C2 P08235 1/20 0.32
GPR88 Q9GZN0 1/20 0.32
CYP2C19 P33261 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
KMT2A Q03164 1/20 0.31
ACE P12821 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1081295 0.93 BACE1 (0.34) BACE1ALDH1A1HPGDTSHRACKR3
SCHEMBL1081296 0.92 BACE1 (0.34) BACE1ALDH1A1HPGDTSHRACKR3
SCHEMBL1081297 0.91 HPGD (0.35) BACE1ALDH1A1HPGDTSHRACKR3
SCHEMBL3696265 0.85 BACE1 (0.34) BACE1ALDH1A1HPGDTSHRACKR3
SCHEMBL3693933 0.85 BACE1 (0.34) BACE1ALDH1A1HPGDTSHRACKR3
SCHEMBL3694157 0.85 LTA4H (0.35) BACE1ALDH1A1HPGDTSHRACKR3
SCHEMBL1193793 0.85 LTA4H (0.35) BACE1ALDH1A1HPGDTSHRACKR3
SCHEMBL1193791 0.85 LTA4H (0.35) BACE1ALDH1A1HPGDTSHRACKR3
SCHEMBL1177679 0.83 HPGD (0.35) BACE1ALDH1A1HPGDTSHRACKR3
SCHEMBL1177677 0.83 HPGD (0.35) BACE1ALDH1A1HPGDTSHRACKR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009127338-A1 OXO-HETEROCYCLIC SUBSTITUTED CARBOXYLIC ACID DERIVATES AND THE USE THEREOF BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2009-10-22 WO disclosed