SCHEMBL4284750

SCHEMBL4284750

CC(C)(C)N(C(=O)c1cccc(O)c1)C(C)(C)C

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.52
CA1 P00915 1/20 0.52
CA2 P00918 1/20 0.52
CA6 P23280 1/20 0.52
CA9 Q16790 1/20 0.52
KDM4E B2RXH2 3/20 0.50
ALDH1A1 P00352 1/20 0.50
PARP1 P09874 1/20 0.50
EGLN2 Q96KS0 1/20 0.47
CYP3A4 P08684 2/20 0.45
CYP2C9 P11712 1/20 0.45
FASN P49327 1/20 0.44
HSD17B1 P14061 5/20 0.44
HSD17B2 P37059 5/20 0.44
GAA P10253 1/20 0.44
MAPT P10636 1/20 0.44
ADRB2 P07550 1/20 0.43
ADRB1 P08588 1/20 0.43
ADRB3 P13945 1/20 0.43
CLK1 P49759 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7898354 0.81 CYP3A4 (0.49) ALDH1A1CYP3A4CYP2C9GAA
SCHEMBL15339830 0.81 HPGD (0.59) PARP1CYP3A4CYP2C9ADRB2ADRB1
SCHEMBL12084828 0.80 CES2 (0.55) KDM4EALDH1A1PARP1CYP3A4CYP2C9
SCHEMBL4277329 0.79 CYP3A4 (0.43) ALDH1A1CYP3A4CYP2C9HSD17B1HSD17B2
SCHEMBL29628546 0.79 CA12 (0.57) CA12CA1CA2CA6CA9
SCHEMBL2645117 0.79 CA12 (0.57) CA12CA1CA2CA6CA9
SCHEMBL11122024 0.78 POLB (0.56) ALDH1A1CYP3A4CYP2C9MAPT
SCHEMBL12084023 0.77 CES2 (0.61) ALDH1A1PARP1HSD17B2ESR1ESR2
SCHEMBL20811957 0.77 MEN1 (0.43) ALDH1A1CYP3A4CYP2C9GAA
SCHEMBL31374707 0.77 CA12 (0.47) CA12CA1CA2CA6CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7608731-B2 Phenylacetic acid compounds ROCHE PALO ALTO LLC (US) 2009-10-27 US disclosed
US-20080108810-A1 Phenylacetic acid compounds ROCHE PALO ALTO LLC 2008-05-08 US disclosed
US-7291729-B2 Process for preparing 3-aryloxy-phenylacetic acid compounds ROCHE PALO ALTO LLC (US) 2007-11-06 US disclosed
EP-1737827-A1 PROCESS FOR PREPARING PYRIDAZINONE COMPOUNDS F.HOFFMANN-LA ROCHE AG (CH) 2007-01-03 EP disclosed
WO-2005100323-A1 PROCESS FOR PREPARING PYRIDAZINONE COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-10-27 WO disclosed
US-20050234236-A1 Process for preparing pyridazinone compounds ROCHE PALO ALTO LLC 2005-10-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080108810-A1 Phenylacetic acid compounds CYP2A6, CYP2B6, DDC CA12 4367/4885CA1 3263/4885CA2 2053/4885
US-20050234236-A1 Process for preparing pyridazinone compounds CYP2A6, CYP2B6, H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16 CA12 4650/4885CA1 4066/4885CA2 3433/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.