SCHEMBL4287009

SCHEMBL4287009

Cn1cncc1C(N)(c1ccc2[nH]c(=O)cc(C(c3cccc(Cl)c3)C3CC3)c2c1)c1ccc(Cl)cn1

nearest known ligand 0.56

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
FNTA P49354 17/20 0.56
FNTB P49356 17/20 0.56
PGGT1B P53609 4/20 0.42
CYP3A4 P08684 3/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3518238 0.89 FNTA (0.56) FNTAFNTBPGGT1BCYP3A4
SCHEMBL4281997 0.79 FNTA (0.60) FNTAFNTBPGGT1BCYP3A4
SCHEMBL4562525 0.72 FNTA (1.00) FNTAFNTBPGGT1BCYP3A4
SCHEMBL4562526 0.72 FNTA (1.00) FNTAFNTBPGGT1BCYP3A4
SCHEMBL6170013 0.71 FNTA (0.82) FNTAFNTBPGGT1B
SCHEMBL3501050 0.70 FNTA (0.84) FNTAFNTBPGGT1BCYP3A4
SCHEMBL28782663 0.70 FNTA (0.72) FNTAFNTBPGGT1BCYP3A4
SCHEMBL2844704 0.70 FNTA (0.72) FNTAFNTBPGGT1BCYP3A4
SCHEMBL6173299 0.69 FNTA (0.82) FNTAFNTBPGGT1BCYP3A4
SCHEMBL3499407 0.69 FNTA (0.71) FNTAFNTBPGGT1BCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009151683-A2 QUINOLINONE FARNESYL TRANSFERASE INHIBITORS FOR THE TREATMENT OF SYNUCLEINOPATHIES AND OTHER INDICATIONS LINK MEDICINE CORPORATION (US) 2009-12-17 WO disclosed