SCHEMBL4288221

SCHEMBL4288221

CC(CCc1nc2c(nc(-c3ccc(F)cc3)n2C)c(=O)[nH]1)C(F)(F)F

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 3/20 0.37
PARP1 P09874 3/20 0.37
ALDH1A1 P00352 3/20 0.36
MAPT P10636 1/20 0.36
DHFR P00374 2/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2C19 P33261 1/20 0.35
KDM4E B2RXH2 2/20 0.35
PDE9A O76083 2/20 0.35
PDE1C Q14123 1/20 0.35
PARP2 Q9UGN5 1/20 0.35
PDE10A Q9Y233 1/20 0.34
ADORA3 P0DMS8 1/20 0.34
ADORA2A P29274 1/20 0.34
ADORA1 P30542 1/20 0.34
KMT2A Q03164 1/20 0.33
ADORA2B P29275 1/20 0.33
LMNA P02545 1/20 0.33
XBP1 P17861 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4774152 0.94 PARP1 (0.38) HPGDPARP1ALDH1A1MAPTDHFR
SCHEMBL4295752 0.91 MEN1 (0.42) HPGDPARP1ALDH1A1MAPTDHFR
SCHEMBL4297801 0.80 PDE9A (0.48) HPGDALDH1A1MAPTDHFRKDM4E
SCHEMBL4296187 0.80 PDE9A (0.48) HPGDALDH1A1MAPTDHFRKDM4E
SCHEMBL4290696 0.79 ALDH1A1 (0.38) HPGDPARP1ALDH1A1MAPTDHFR
SCHEMBL4292483 0.78 PDE9A (0.36) HPGDPARP1ALDH1A1DHFRKDM4E
SCHEMBL4767017 0.76 POLB (0.40) HPGDPARP1ALDH1A1MAPTDHFR
SCHEMBL4769038 0.74 MEN1 (0.44) HPGDPARP1ALDH1A1MAPTDHFR
SCHEMBL4776971 0.73 MEN1 (0.46) HPGDPARP1ALDH1A1MAPTDHFR
SCHEMBL4290740 0.72 MEN1 (0.42) HPGDALDH1A1MAPTDHFRKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2061470-A2 HALOALKYL-SUBSTITUTED PYRIMIDINONE DERIVATIVES Neurogen Corporation (US) 2009-05-27 EP claimed
WO-2008024433-A2 HALOALKYL-SUBSTITUTED PYRIMIDINONE DERIVATIVES NEUROGEN CORPORATION (US) 2008-02-28 WO claimed