SCHEMBL4290696

SCHEMBL4290696

CCn1c(-c2ccc(Cl)cc2)nc2c(=O)[nH]c(CCC(C)C(F)(F)F)nc21

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.38
KDM4E B2RXH2 4/20 0.38
HPGD P15428 4/20 0.38
PKM P14618 1/20 0.38
PDE9A O76083 2/20 0.37
PDE1C Q14123 1/20 0.37
TDP1 Q9NUW8 2/20 0.37
LMNA P02545 1/20 0.37
GFER P55789 1/20 0.37
APOBEC3G Q9HC16 1/20 0.37
KMT2A Q03164 5/20 0.34
MEN1 O00255 4/20 0.34
HTT P42858 2/20 0.34
POLB P06746 1/20 0.34
TRPV1 Q8NER1 1/20 0.34
DHFR P00374 1/20 0.34
MAPT P10636 1/20 0.33
PDE10A Q9Y233 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
PARP1 P09874 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4292483 0.91 PDE9A (0.36) ALDH1A1KDM4EHPGDPKMPDE9A
SCHEMBL4295752 0.88 MEN1 (0.42) ALDH1A1KDM4EHPGDPKMPDE9A
SCHEMBL4774602 0.85 ALDH1A1 (0.42) ALDH1A1KDM4EHPGDPKMTDP1
SCHEMBL4776139 0.84 ALDH1A1 (0.41) ALDH1A1KDM4EHPGDPKMTDP1
SCHEMBL4768853 0.83 ALDH1A1 (0.43) ALDH1A1KDM4EHPGDPKMTDP1
SCHEMBL4774287 0.83 ALDH1A1 (0.41) ALDH1A1KDM4EHPGDPKMTDP1
SCHEMBL4772661 0.81 ALDH1A1 (0.44) ALDH1A1KDM4EHPGDPKMTDP1
SCHEMBL4290620 0.80 PDE9A (0.45) ALDH1A1KDM4EHPGDPKMPDE9A
SCHEMBL4297747 0.79 PDE9A (0.46) ALDH1A1KDM4EHPGDPDE9APDE1C
SCHEMBL4288221 0.79 HPGD (0.37) ALDH1A1KDM4EHPGDPDE9APDE1C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2061470-A2 HALOALKYL-SUBSTITUTED PYRIMIDINONE DERIVATIVES Neurogen Corporation (US) 2009-05-27 EP claimed
WO-2008024433-A2 HALOALKYL-SUBSTITUTED PYRIMIDINONE DERIVATIVES NEUROGEN CORPORATION (US) 2008-02-28 WO claimed