SCHEMBL4295294

SCHEMBL4295294

CCOC(=O)c1cc(C#N)c(N2CCNCC2)nc1CF

nearest known ligand 0.73

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.73
KDM4E B2RXH2 5/20 0.55
L3MBTL1 Q9Y468 4/20 0.55
LMNA P02545 1/20 0.55
HPGD P15428 1/20 0.55
TDP1 Q9NUW8 1/20 0.55
MEN1 O00255 2/20 0.53
KMT2A Q03164 2/20 0.53
MAPT P10636 1/20 0.53
P2RY12 Q9H244 12/20 0.50
HTT P42858 1/20 0.49
NPSR1 Q6W5P4 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4425610 0.89 ALDH1A1 (0.75) ALDH1A1KDM4EL3MBTL1LMNAHPGD
SCHEMBL3874439 0.87 ALDH1A1 (0.76) ALDH1A1KDM4EL3MBTL1LMNAHPGD
SCHEMBL30999840 0.87 ALDH1A1 (0.76) ALDH1A1KDM4EL3MBTL1LMNAHPGD
Hydrochloric Acid SCHEMBL4878714 0.86 ALDH1A1 (0.74) ALDH1A1KDM4EL3MBTL1LMNAHPGD
SCHEMBL3581873 0.85 P2RY12 (0.56) ALDH1A1KDM4EL3MBTL1LMNAHPGD
SCHEMBL30999844 0.84 ALDH1A1 (1.00) ALDH1A1KDM4EP2RY12NPSR1
SCHEMBL3926740 0.84 ALDH1A1 (1.00) ALDH1A1KDM4EP2RY12NPSR1
SCHEMBL4425609 0.84 ALDH1A1 (0.84) ALDH1A1KDM4EP2RY12NPSR1
SCHEMBL4005299 0.83 ALDH1A1 (0.70) ALDH1A1KDM4EL3MBTL1LMNAHPGD
SCHEMBL14598715 0.83 ALDH1A1 (0.69) ALDH1A1KDM4EL3MBTL1LMNAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2041111-A1 NEW PYRIDINE ANALOGUES AstraZeneca AB (SE) 2009-04-01 EP disclosed
WO-2008002247-A1 NEW PYRIDINE ANALOGUES ASTRAZENECA AB (SE) 2008-01-03 WO disclosed