SCHEMBL4425609

SCHEMBL4425609

CCOC(=O)c1cc(C#N)c(N2CCNCC2)nc1C(F)(F)CF

nearest known ligand 0.84

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.84
P2RY12 Q9H244 17/20 0.58
KDM4E B2RXH2 1/20 0.56
NPSR1 Q6W5P4 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3926740 0.91 ALDH1A1 (1.00) ALDH1A1P2RY12KDM4ENPSR1
SCHEMBL30999844 0.91 ALDH1A1 (1.00) ALDH1A1P2RY12KDM4ENPSR1
SCHEMBL4295294 0.84 ALDH1A1 (0.73) ALDH1A1P2RY12KDM4ENPSR1
SCHEMBL3874439 0.84 ALDH1A1 (0.76) ALDH1A1P2RY12KDM4E
SCHEMBL30999840 0.84 ALDH1A1 (0.76) ALDH1A1P2RY12KDM4E
SCHEMBL4425610 0.83 ALDH1A1 (0.75) ALDH1A1P2RY12KDM4ENPSR1
Hydrochloric Acid SCHEMBL4878714 0.83 ALDH1A1 (0.74) ALDH1A1P2RY12KDM4E
SCHEMBL5066024 0.82 ALDH1A1 (0.83) ALDH1A1P2RY12KDM4ENPSR1
SCHEMBL5423936 0.81 ALDH1A1 (0.56) ALDH1A1P2RY12KDM4ENPSR1
SCHEMBL4005299 0.80 ALDH1A1 (0.70) ALDH1A1P2RY12KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2041111-A1 NEW PYRIDINE ANALOGUES AstraZeneca AB (SE) 2009-04-01 EP disclosed
WO-2008002247-A1 NEW PYRIDINE ANALOGUES ASTRAZENECA AB (SE) 2008-01-03 WO disclosed