SCHEMBL4296010

SCHEMBL4296010

CN(C)CCOc1ccc(-c2cccc(N)n2)c(O)c1.COc1cc(OCC(N)=O)ccc1-c1cccc(N)n1

nearest known ligand 0.57

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 14/20 0.57
NOS3 P29474 9/20 0.57
NOS2 P35228 6/20 0.49
ACACA Q13085 1/20 0.41
CHRNB2 P17787 1/20 0.41
CHRNA4 P43681 1/20 0.41
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
HSP90B1 P14625 1/20 0.39
TRAP1 Q12931 1/20 0.39
MEN1 O00255 1/20 0.39
LMNA P02545 1/20 0.39
MAPT P10636 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL218649 0.97 NOS1 (0.54) NOS1NOS3NOS2ACACACHRNB2
SCHEMBL218712 0.88 NOS1 (0.65) NOS1NOS3NOS2CHRNB2CHRNA4
SCHEMBL6585074 0.87 ACACA (0.50) NOS1NOS3ACACAKDM4EMEN1
SCHEMBL222693 0.87 NOS1 (0.73) NOS1NOS3NOS2CHRNB2CHRNA4
Guaiacol SCHEMBL4699468 0.86 NOS1 (0.62) NOS1NOS3NOS2CHRNB2CHRNA4
SCHEMBL6585604 0.85 NOS1 (0.61) NOS1NOS3NOS2CHRNB2CHRNA4
SCHEMBL4692515 0.84 NOS1 (0.60) NOS1NOS3NOS2CHRNB2CHRNA4
SCHEMBL220285 0.78 NOS1 (0.61) NOS1NOS3NOS2CHRNB2CHRNA4
SCHEMBL220827 0.77 NOS1 (0.63) NOS1NOS3NOS2
SCHEMBL4282766 0.77 NOS1 (0.53) NOS1NOS3NOS2KDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009158646-A1 THERAPEUTIC COMPUNDS AND RELATED METHODS OF USE ELIXIR PHARMACEUTICALS, INC. (US) 2009-12-30 WO disclosed