SCHEMBL4298066

SCHEMBL4298066

COc1cc(N)c2c(c1)CC(CO)O2

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.37
ALDH1A1 P00352 3/20 0.37
HPGD P15428 1/20 0.37
HRH3 Q9Y5N1 2/20 0.36
PRKAB2 O43741 1/20 0.35
PRKAG1 P54619 1/20 0.35
PRKAA2 P54646 1/20 0.35
PRKAA1 Q13131 1/20 0.35
PRKAG3 Q9UGI9 1/20 0.35
PRKAG2 Q9UGJ0 1/20 0.35
PRKAB1 Q9Y478 1/20 0.35
RXFP1 Q9HBX9 1/20 0.33
GAA P10253 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
MEN1 O00255 2/20 0.33
MAPT P10636 2/20 0.33
THRB P10828 2/20 0.33
KMT2A Q03164 2/20 0.33
RECQL P46063 1/20 0.33
BLM P54132 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13056378 0.84 KDM4E (0.43) KDM4EALDH1A1HPGDHRH3PRKAB2
SCHEMBL15667032 0.80 RXFP1 (0.37) KDM4EALDH1A1HPGDRXFP1GAA
SCHEMBL4236397 0.80 CA1 (0.42) KDM4EALDH1A1HPGDHRH3PRKAB2
SCHEMBL10044954 0.79 HRH3 (0.38) KDM4EALDH1A1HPGDHRH3PRKAB2
SCHEMBL4294701 0.77 MTNR1A (0.39) KDM4EALDH1A1HPGDGAASMN1; SMN2
SCHEMBL4290552 0.74 MTNR1A (0.39) KDM4EALDH1A1GAAMEN1MAPT
SCHEMBL18167170 0.72 PIK3CG (0.42)
SCHEMBL15758336 0.71 KDM4E (0.42) KDM4EALDH1A1HPGDPRKAB2PRKAG1
SCHEMBL7288132 0.70 HRH3 (0.49) HRH3DRD2DRD3ACHE
SCHEMBL7288140 0.70 HRH3 (0.49) HRH3DRD2DRD3ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2630129-B1 QUINOXALINE DERIVATES MERCK PATENT GMBH (DE) 2016-10-26 EP disclosed
WO-2012052102-A1 QUINOXALINE DERIVATES MERCK PATENT GMBH (DE) 2012-04-26 WO disclosed