SCHEMBL7288140

SCHEMBL7288140

COc1ccc2c(c1)O[C@@H](CO)C2

nearest known ligand 0.53

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 2/20 0.49
FFAR1 O14842 1/20 0.42
MTNR1A P48039 1/20 0.42
CA2 P00918 1/20 0.40
CA5A P35218 1/20 0.40
CYP19A1 P11511 4/20 0.40
MAOB P27338 2/20 0.40
CYP3A4 P08684 1/20 0.40
ACHE P22303 1/20 0.39
DRD2 P14416 1/20 0.39
DRD3 P35462 1/20 0.39
GABRA1 P14867 1/20 0.39
GABRB2 P47870 1/20 0.39
HTR1A P08908 1/20 0.38
HTR1D P28221 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7288132 1.00 HRH3 (0.49) HRH3FFAR1MTNR1ACA2CA5A
SCHEMBL7317620 0.85 FFAR1 (0.54) FFAR1CA2CA5ACYP3A4DRD2
SCHEMBL7317624 0.85 FFAR1 (0.54) FFAR1CA2CA5ACYP3A4DRD2
SCHEMBL4234794 0.84 HRH3 (0.49) HRH3FFAR1MTNR1ACA2CA5A
SCHEMBL17761390 0.81 HRH3 (0.44) HRH3FFAR1MTNR1ACA2CA5A
SCHEMBL177102 0.78 CYP26A1 (0.47) HRH3FFAR1CYP19A1
SCHEMBL15447319 0.78 ELANE (0.43) FFAR1MTNR1ACA2CA5A
SCHEMBL177299 0.77 FFAR1 (0.39) HRH3FFAR1MTNR1ACYP3A4
SCHEMBL1870686 0.77 MTNR1A (0.63) FFAR1MTNR1A
SCHEMBL11484008 0.77 MTNR1A (0.56) FFAR1MTNR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6359138-B1 CENTRAL NERVOUS SYSTEM DISORDERS HOFFMANN-LA ROCHE INC. 2002-03-19 US disclosed
EP-0846683-B1 4-Hydroxy-piperidine derivatives HOFFMANN LA ROCHE (CH) 2001-09-19 EP disclosed
EP-0846683-A1 4-Hydroxy-piperidine derivatives F. HOFFMANN-LA ROCHE AG (CH) 1998-06-10 EP disclosed