SCHEMBL4304368

SCHEMBL4304368

NC(=O)CCCCc1cccnc1

nearest known ligand 0.76

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TBXAS1 P24557 8/20 0.76
HRH1 P35367 2/20 0.62
CYP2A6 P11509 1/20 0.61
TDP1 Q9NUW8 1/20 0.59
L3MBTL1 Q9Y468 1/20 0.59
RECQL P46063 1/20 0.58
CHRNA7 P36544 1/20 0.55
MAPT P10636 1/20 0.54
NAPRT Q6XQN6 1/20 0.51
CYP3A4 P08684 2/20 0.51
CYP1A2 P05177 1/20 0.50
CYP2C9 P11712 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18248629 0.98 TBXAS1 (0.77) TBXAS1HRH1CYP2A6TDP1L3MBTL1
SCHEMBL14959999 0.98 TBXAS1 (0.77) TBXAS1HRH1CYP2A6TDP1L3MBTL1
SCHEMBL10772829 0.98 TBXAS1 (0.77) TBXAS1HRH1CYP2A6TDP1L3MBTL1
SCHEMBL933853 0.95 TBXAS1 (0.68) TBXAS1HRH1CYP2A6TDP1L3MBTL1
SCHEMBL18248504 0.90 TBXAS1 (0.65) TBXAS1HRH1CYP2A6TDP1L3MBTL1
SCHEMBL18248608 0.90 TBXAS1 (0.65) TBXAS1HRH1CYP2A6TDP1L3MBTL1
SCHEMBL83186 0.89 RECQL (0.62) TBXAS1HRH1CYP2A6RECQLCHRNA7
Hydrochloric Acid SCHEMBL5349530 0.88 TBXAS1 (0.61) TBXAS1HRH1CYP2A6RECQLCHRNA7
SCHEMBL18248525 0.87 TBXAS1 (0.62) TBXAS1HRH1CYP2A6RECQLMAPT
SCHEMBL744045 0.86 TBXAS1 (1.00) TBXAS1HRH1CYP2A6TDP1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009126675-A1 2-SULFONYLAMINO-4-HETEROARYL BUTYRAMIDE ANTAGONISTS OF CCR10 BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-10-15 WO disclosed
US-4551460-A ANTICOAGULANTS, CARDIOVASCULAR DISORDERS HOFFMANN-LA ROCHE INC. (US) 1985-11-05 US disclosed