SCHEMBL4304834

SCHEMBL4304834

CC(O)Cc1ccc2nc(C#N)ccc2c1

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NQO1 P15559 1/20 0.51
HRH3 Q9Y5N1 2/20 0.39
SCN9A Q15858 6/20 0.39
HTR2A P28223 1/20 0.34
HTR2C P28335 1/20 0.34
HTR2B P41595 1/20 0.34
TTR P02766 2/20 0.34
SOS2 Q07890 1/20 0.33
CTSK P43235 1/20 0.33
ALDH1A1 P00352 2/20 0.33
HPGDS O60760 1/20 0.33
ALOX15 P16050 1/20 0.33
KDM4E B2RXH2 1/20 0.32
TSHR P16473 1/20 0.32
CASP1 P29466 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15047212 0.80 NQO1 (0.58) NQO1HRH3TTRCTSKALDH1A1
SCHEMBL17442633 0.80 NQO1 (0.54) NQO1SCN9ATTRSOS2CTSK
SCHEMBL16881222 0.76 NQO1 (0.54) NQO1HRH3TTRSOS2CTSK
SCHEMBL17442652 0.76 NQO1 (0.54) NQO1HRH3TTRSOS2CTSK
SCHEMBL9176689 0.75 HTR2A (0.53) HRH3HTR2AHTR2CHTR2BTTR
SCHEMBL25401591 0.75 NQO1 (0.49) NQO1ALDH1A1KDM4ETSHR
SCHEMBL4301102 0.73 MGAM (0.46) SCN9AALDH1A1KDM4E
SCHEMBL1688377 0.73 NQO1 (0.58) NQO1SCN9ATTRSOS2CTSK
SCHEMBL6843917 0.73 HTR2A (0.52) HTR2AHTR2CHTR2BTTRALDH1A1
SCHEMBL21639257 0.71 CTSS (0.57) CTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2024272-A2 AMIDE DERIVATIVES AS ION-CHANNEL LIGANDS AND PHARMACEUTICAL COMPOSITIONS AND METHODS OF USING THE SAME Renovis, Inc. (US) 2009-02-18 EP disclosed
WO-2007133637-A2 AMIDE DERIVATIVES AS ION-CHANNEL LIGANDS AND PHARMACEUTICAL COMPOSITIONS AND METHODS OF USING THE SAME RENOVIS, INC. (US) 2007-11-22 WO disclosed