Indene

Indene

SCHEMBL4305388

C1=Cc2ccccc2C1.C1=Cc2ccccc2C1.[Zr]c1cc2ccccc2[nH]1

nearest known ligand 0.36

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.36
CA2 P00918 2/20 0.36
AOC3 Q16853 2/20 0.36
BRD4 O60885 1/20 0.36
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
KDM4E B2RXH2 2/20 0.33
MAPT P10636 2/20 0.33
ALDH1A1 P00352 2/20 0.33
LOXL2 Q9Y4K0 1/20 0.33
FLT3 P36888 1/20 0.33
CYP2A6 P11509 1/20 0.33
HRH4 Q9H3N8 2/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C19 P33261 1/20 0.33
AURKA O14965 1/20 0.33
KDR P35968 1/20 0.33
DAO P14920 2/20 0.33
HPGD P15428 1/20 0.33
SRD5A2 P31213 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Indene SCHEMBL6247868 1.00 CA1 (0.36) CA1CA2AOC3BRD4NPC1
Indene SCHEMBL6627120 0.81 CA1 (0.36) CA1CA2AOC3BRD4NPC1
Indene SCHEMBL6628425 0.81 CA2 (0.36) CA1CA2AOC3BRD4NPC1
SCHEMBL7644722 0.78 AOC3 (0.54) CA1CA2AOC3BRD4NPC1
Indene SCHEMBL4452296 0.76 NPC1 (0.33) CA1CA2AOC3BRD4NPC1
Anthracene SCHEMBL28057537 0.76 CA1 (0.47) CA1CA2MAPTALDH1A1CYP2D6
Naphthalene SCHEMBL2783692 0.76 CA1 (0.50) CA1CA2CYP2A6CYP2D6CYP2C19
SCHEMBL5071409 0.76 LOXL2 (0.42) CA1AOC3BRD4NPC1RAB9A
SCHEMBL5071399 0.76 LOXL2 (0.42) CA1AOC3BRD4NPC1RAB9A
Indene SCHEMBL4756119 0.74 AHR (0.59) CA1CA2NPC1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 19 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8475898-B2 Polyolefin resin blends for crack-resistant pipe EQUISTAR CHEMICALS, LP (US) 2013-07-02 US disclosed
EP-1567561-B1 BIMETALLIC INDENOINDOLYL CATALYSTS EQUISTAR CHEM LP (US) 2009-05-27 EP disclosed
WO-2009032049-A1 OLEFIN POLYMERIZATION PROCESS EQUISTAR CHEMICALS, LP (US) 2009-03-12 WO disclosed
US-20090061135-A1 Polyolefin resin blends for crack-resistant pipe EQUISTAR CHEMICALS, LP 2009-03-05 US disclosed
EP-1567561-A1 BIMETALLIC INDENOINDOLYL CATALYSTS Equistar Chemicals, LP (US) 2005-08-31 EP disclosed
US-6908972-B2 Method for making polyolefins EQUISTAR CHEMICALS, LP (US) 2005-06-21 US disclosed
EP-1509554-A1 HIGH-TEMPERATURE OLEFIN POLYMERISATION PROCESS IN SOLUTION Equistar Chemicals, LP (US) 2005-03-02 EP disclosed
EP-1497343-A1 METHOD FOR POLYMERISATION OF OLEFINS WITH INDENO-INDOLYL CATALYSTS Equistar Chemicals, LP (US) 2005-01-19 EP disclosed
US-6841500-B2 Bimetallic indenoindolyl catalysts EQUISTAR CHEMICALS, LP (US) 2005-01-11 US disclosed
US-6756455-B2 POLYMERIZING OLEFINS IN SOLUTION IN MULTISTAGE REACTOR UNDER ADIABATIC CONDITIONS AT SPECIFIED TEMPERATURE AND PRESSURE IN PRESENCE OF CATALYST SYSTEM INCLUDING ACTIVATOR AND COMPLEX COMPRISING TRANSITION METAL AND BRIDGED INDENOINDOLYL LIGAND EQUISTAR CHEMICALS, LP 2004-06-29 US disclosed
WO-2004050718-A1 BIMETALLIC INDENOINDOLYL CATALYSTS EQUISTAR CHEMICALS, LP (US) 2004-06-17 WO disclosed
US-20040106514-A1 Bimetallic indenoindolyl catalysts EQUISTAR CHEMICALS, LP 2004-06-03 US disclosed
EP-1417031-A1 AMINE ELIMINATION PROCESS FOR MAKING SINGLE-SITE CATALYSTS Equistar Chemicals, LP (US) 2004-05-12 EP disclosed
WO-2003102042-A1 HIGH-TEMPERATURE OLEFIN POLYMERISATION PROCESS IN SOLUTION EQUISTAR CHEMICALS, LP (US) 2003-12-11 WO disclosed
US-20030229188-A1 High-temperature solution process for polyolefin manufacture EQUISTAR CHEMICALS, LP 2003-12-11 US disclosed
WO-2003089485-A1 METHOD FOR POLYMERISATION OF OLEFINS WITH INDENO-INDOLYL CATALYSTS EQUISTAR CHEMICALS, LP (US) 2003-10-30 WO disclosed
US-20030195306-A1 Method for making polyolefins EQUISTAR CHEMICALS, LP 2003-10-16 US disclosed
WO-2003015917-A1 AMINE ELIMINATION PROCESS FOR MAKING SINGLE-SITE CATALYSTS EQUISTAR CHEMICALS, LP (US) 2003-02-27 WO disclosed
US-6440889-B1 OLEFIN POLYMERIZATION CATALYSTS; GROUP 4 METAL COMPLEXES WITH SINGLE ANIONIC INDENOINDOLYL LIGAND; REACTING AN INDENOINDOLE WITH TETRAKIS(DIALKYLAMINO) ZIRCONIUM COMPOUND; HALOGENATING; REACTING WITH A CYCLOPENTADIENYL ANION EQUISTAR CHEMICALS, LP 2002-08-27 US disclosed