SCHEMBL4306583

SCHEMBL4306583

CCOC(=O)c1cn(C2CC2)c2cc(F)c(F)cc2c1=O

nearest known ligand 0.73

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.60
ADRB2 P07550 1/20 0.56
KDM4E B2RXH2 5/20 0.54
ALDH1A1 P00352 5/20 0.54
HPGD P15428 5/20 0.54
HSD17B10 Q99714 4/20 0.54
LMNA P02545 3/20 0.54
MAPT P10636 1/20 0.54
TOP2A P11388 2/20 0.49
TOP2B Q02880 2/20 0.49
CYP1A2 P05177 1/20 0.49
CYP2C9 P11712 1/20 0.49
STAT3 P40763 1/20 0.45
KCNH2 Q12809 1/20 0.43
PIK3CD O00329 1/20 0.43
PIK3R1 P27986 1/20 0.43
PIK3CA P42336 1/20 0.43
PIK3CG P48736 1/20 0.43
HTT P42858 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29576844 1.00 KMT2A (0.60) KMT2AADRB2KDM4EALDH1A1HPGD
SCHEMBL10577000 0.92 KMT2A (0.54) KMT2AADRB2KDM4EALDH1A1HPGD
SCHEMBL29475787 0.91 ADRB2 (0.53) KMT2AADRB2KDM4EALDH1A1HPGD
SCHEMBL7889777 0.91 ADRB2 (0.53) KMT2AADRB2KDM4EALDH1A1HPGD
SCHEMBL7579219 0.91 ADRB2 (0.53) KMT2AADRB2KDM4EALDH1A1HPGD
SCHEMBL22795687 0.91 KDM4E (0.53) KMT2AADRB2KDM4EALDH1A1HPGD
SCHEMBL9442762 0.90 ADRB2 (0.52) KMT2AADRB2KDM4EALDH1A1HPGD
SCHEMBL9260574 0.90 KMT2A (0.57) KMT2AADRB2KDM4EALDH1A1HPGD
SCHEMBL9270695 0.90 KMT2A (0.57) KMT2AADRB2KDM4EALDH1A1HPGD
SCHEMBL1243388 0.88 KMT2A (0.53) KMT2AADRB2KDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 82 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116283766-A Cyanomethyl quinolone compound and preparation method and application thereof 西南大学 2023-06-23 CN claimed
CN-115636785-A Quinolone cyanoacetate compounds and pharmaceutically acceptable salts thereof, and preparation method and application thereof 西南大学 2023-01-24 CN claimed
JP-9309880-A None JP disclosed
US-20250313561-A1 NEXT-GENERATION MODULATORS OF STIMULATOR OF INTERFERON GENES (STING) RYVU THERAPEUTICS S A (PL) 2025-10-09 US disclosed
EP-3630779-B1 ANTIBIOTIC RESISTANCE BREAKERS KING S COLLEGE LONDON (GB) 2025-09-03 EP disclosed
US-12344606-B2 Next-generation modulators of stimulator of interferon genes (STING) Ryvu Therapeutics S.A. (PL) 2025-07-01 US disclosed
CN-115636785-B Quinolone cyanoacetate compound and pharmaceutically acceptable salt thereof, and preparation method and application thereof 西南大学 2024-05-28 CN disclosed
CN-117486796-A Synthesis method of key intermediate of quinolone antibacterial drug 山东京新药业有限公司 2024-02-02 CN disclosed
EP-3983078-B1 NEXT-GENERATION MODULATORS OF STIMULATOR OF INTERFERON GENES (STING) RYVU THERAPEUTICS S A (PL) 2023-11-15 EP disclosed
EP-3983078-B1 NEXT-GENERATION MODULATORS OF STIMULATOR OF INTERFERON GENES (STING) RYVU THERAPEUTICS S A (PL) 2023-11-15 EP disclosed
US-11746116-B2 Antibiotic resistance breakers KING'S COLLEGE LONDON (GB) 2023-09-05 US disclosed
US-4956465-A Bactericides BAYER AKTIENGESELLSCHAFT (DE) 1990-09-11 US disclosed
US-4920120-A 3-CARBOXY, 4-OXO, 6-FLUORO, 7-NITROGEN-CONTAINING RING 1,4-DIHYDRO-1,8-NAPHTHYRIDINES WARNER-LAMBERT COMPANY (US) 1990-04-24 US disclosed
EP-0342849-A2 Intermediates for preparing 1,4-dihydro-4-oxo-quinoline-3-carboxylic acid esters PFIZER INC. (US) 1989-11-23 EP disclosed
US-4880814-A 7-cycloalkyl naphthyridines ABBOTT LABORATORIES (US) 1989-11-14 US disclosed
EP-0326891-A2 Antibacterial agents WARNER-LAMBERT COMPANY (US) 1989-08-09 EP disclosed
WO-1989006649-A2 ANTIBACTERIAL AGENTS WARNER-LAMBERT COMPANY (US) 1989-07-27 WO disclosed
US-4820716-A ANIMAL GROWTH REGULATORS, BACTERICIDES BAYER AKTIENGESELLSCHAFT (DE) 1989-04-11 US disclosed
US-4599334-A 7-(3-aryl-1-piperazinyl)- and 7-(3-cyclohexyl-1-piperazinyl)-3-quinolonecarboxylic acid antibacterials BAYER AKTIENGESELLSCHAFT (DE) 1986-07-08 US disclosed
US-4588726-A 1-cyclopropyl-6-fluoro-1,4-dihydro-4-oxo-7-(3-oxo-1-piperazinyl)-3-quinolinecarboxylic acid antibacterial agents BAYER AKTIENGESELLSCHAFT (DE) 1986-05-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12344606-B2 Next-generation modulators of stimulator of interferon genes (STING) STING1, IRF3, CGAS KMT2A 4634/4885ADRB2 214/4885KDM4E 4160/4885
US-11746116-B2 Antibiotic resistance breakers ABCC1, ARL1, AKR1C3 KMT2A 4080/4885ADRB2 1179/4885KDM4E 3599/4885
US-20250313561-A1 NEXT-GENERATION MODULATORS OF STIMULATOR OF INTERFERON GENES (STING) STING1, IRF3, CGAS KMT2A 4634/4885ADRB2 214/4885KDM4E 4160/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.