SCHEMBL43092

SCHEMBL43092

NP(N)(=O)ON1CCOCC1

nearest known ligand 0.35

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MMP1 P03956 1/20 0.35
MMP3 P08254 1/20 0.35
MMP8 P22894 1/20 0.35
ANPEP P15144 1/20 0.34
CA12 O43570 1/20 0.32
CA7 P43166 1/20 0.32
CA14 Q9ULX7 1/20 0.32
MAPT P10636 1/20 0.31
KDM4E B2RXH2 2/20 0.31
GAA P10253 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1615660 0.86 MMP1 (0.35) MMP1MMP3MMP8ANPEPCA12
SCHEMBL1615661 0.82 MMP1 (0.42) MMP1MMP3MMP8ANPEPCA12
SCHEMBL18426999 0.82 MMP1 (0.33) MMP1MMP3MMP8ANPEPCA12
SCHEMBL21145497 0.80 MMP1 (0.41) MMP1MMP3MMP8ANPEPCA12
SCHEMBL4302310 0.80 MMP1 (0.38) MMP1MMP3MMP8ANPEPCA12
SCHEMBL28308289 0.79 MMP1 (0.31) MMP1MMP3MMP8ANPEP
SCHEMBL27667273 0.77 MMP1 (0.33) MMP1MMP3MMP8ANPEPCA12
SCHEMBL329844 0.76 MMP1 (0.45) MMP1MMP3MMP8ANPEPCA12
SCHEMBL8505349 0.76 TSHR (0.36) MMP1MMP3MMP8ANPEPCA12
SCHEMBL2974387 0.76 MMP1 (0.45) MMP1MMP3MMP8ANPEPCA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 5699 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4291244-B1 CELL-PENETRATING PEPTIDE CONJUGATES AND METHODS OF THEIR USE UNIV OXFORD INNOVATION LTD (GB) 2025-12-10 EP claimed
EP-3250591-B1 HUMAN ANTIBODIES TO EBOLA VIRUS GLYCOPROTEIN REGENERON PHARMA (US) 2025-11-12 EP claimed
US-20250332270-A1 Targeting Skin-Related Conditions Using Bottlebrush Polymer-Conjugated Oligonucleotides UNIV NORTHEASTERN (US) 2025-10-30 US claimed
EP-4610278-A2 TARGETED SAPONIN-NUCLEIC ACID CONJUGATES FOR TREATMENT OF MUSCLE WASTING DISORDERS Sapreme Technologies B.V. (NL) 2025-09-03 EP claimed
US-20250250564-A2 COMPOSITIONS COMPRISING THERAPEUTIC NUCLEIC ACID AND SAPONIN FOR THE TREATMENT OF MUSCLE-WASTING DISORDERS SAPREME TECH BV (NL) 2025-08-07 US claimed
EP-4452331-B1 TARGETED SAPONIN-NUCLEIC ACID CONJUGATES FOR TREATMENT OF MUSCLE WASTING DISORDERS SAPREME TECH BV (NL) 2025-08-06 EP claimed
US-20250163418-A1 Brush polymer-oligonucleotide conjugates for the treatment of muscular dystrophy UNIV NORTHEASTERN (US) 2025-05-22 US claimed
WO-2025085618-A1 METHODS FOR APPENDING ADAPTORS ONTO POLYNUCLEOTIDES ILLUMINA, INC. (US) 2025-04-24 WO claimed
EP-3660154-B1 ANTISENSE NUCLEIC ACID FOR USE IN TREATING DUCHENNE MUSCULAR DYSTROPHY NIPPON SHINYAKU CO LTD (JP) 2025-04-16 EP claimed
US-20250082759-A1 COMPOSITIONS COMPRISING THERAPEUTIC NUCLEIC ACID AND TARGETED SAPONIN FOR THE TREATMENT OF MUSCLE-WASTING DISORDERS SAPREME TECHNOLOGIES B.V. (NL) 2025-03-13 US claimed
US-20060147952-A1 2'-O-methyl-phosphorothioate oligoribonucleotide modification; peptide nucleic acids, locked nucleic acids, and/or morpholino phosphorodiamidate oligonucleotides; splicing to skip hybridization ACADEMISCH ZIEKENHUIS LEIDEN (NL) 2006-07-06 US claimed
US-20060099616-A1 2'-O-methyl-phosphorothioate oligoribonucleotide modification; peptide nucleic acids, locked nucleic acids, and/or morpholino phosphorodiamidate oligonucleotides; splicing to skip hybridization ACADEMISCH ZIEKENHUIS LEIDEN (NL) 2006-05-11 US claimed
WO-2006002540-A1 OLIGONUCLEOTIDES TARGETING PRION DISEASES AND USES REPLICOR INC. (CA) 2006-01-12 WO claimed
EP-1606407-A2 MODULATION OF EXON RECOGNITION IN PRE-MRNA BY INTERFERING WITH THE SECONDARY RNA STRUCTURE Academisch Ziekenhuis Leiden (NL) 2005-12-21 EP claimed
US-20050233455-A1 Acyclic linker-containing oligonucleotides and uses thereof DAMHA MASAD J 2005-10-20 US claimed
WO-2004083432-A1 MODULATION OF EXON RECOGNITION IN PRE-MRNA BY INTERFERING WITH THE SECONDARY RNA STRUCTURE ACADEMISCH ZIEKENHUIS LEIDEN (NL) 2004-09-30 WO claimed
WO-2004083446-A2 MODULATION OF EXON RECOGNITION IN PRE-MRNA BY INTERFERING WITH THE SECONDARY RNA STRUCTURE ACADEMISCH ZIEKENHUIS LEIDEN (NL) 2004-09-30 WO claimed
EP-1440079-A1 ACYCLIC LINKER-CONTAINING OLIGONUCLEOTIDES AND USES THEREOF McGILL UNIVERSITY (CA) 2004-07-28 EP claimed
US-20030220249-A1 Factors for angiogenesis, vasculogenesis, cartilage formation, bone formation, and methods of use thereof DISCOVERY GENOMICS, INC. 2003-11-27 US claimed
WO-2003037909-A1 ACYCLIC LINKER-CONTAINING OLIGONUCLEOTIDES AND USES THEREOF MCGILL UNIVERSITY (CA) 2003-05-08 WO claimed