SCHEMBL4316385

SCHEMBL4316385

Cc1c(C(=O)O)c2cc(=O)cc(F)c-2cn1-c1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
ABCB1 P08183 1/20 0.40
NOTUM Q6P988 5/20 0.39
MAPK1 P28482 1/20 0.37
GAA P10253 1/20 0.36
GFER P55789 1/20 0.36
ALDH1A1 P00352 2/20 0.35
COMT P21964 1/20 0.35
KDM4E B2RXH2 3/20 0.35
CYP1A2 P05177 1/20 0.35
HPGD P15428 1/20 0.35
BLM P54132 1/20 0.35
HSD17B10 Q99714 1/20 0.35
ATM Q13315 1/20 0.34
LMNA P02545 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3632665 0.91 ABCB1 (0.50) MEN1KMT2AABCB1NOTUMALDH1A1
SCHEMBL3633358 0.90 NOTUM (0.44) MEN1KMT2AABCB1NOTUMALDH1A1
SCHEMBL1551329 0.88 AKR1C3 (0.37) MEN1KMT2AABCB1LMNA
SCHEMBL3634622 0.87 NOTUM (0.45) MEN1KMT2ANOTUMKDM4EATM
SCHEMBL3634031 0.87 PLA2G4A (0.35) MEN1KMT2AMAPK1
SCHEMBL3632614 0.86 MEN1 (0.45) MEN1KMT2AABCB1NOTUMMAPK1
SCHEMBL3629049 0.84 MEN1 (0.43) MEN1KMT2AABCB1NOTUMMAPK1
SCHEMBL1032110 0.84 MEN1 (0.43) MEN1KMT2AABCB1NOTUMMAPK1
SCHEMBL1550103 0.83 SMN1; SMN2 (0.39) MEN1KMT2AGAAKDM4ELMNA
SCHEMBL4284158 0.82 ABCB1 (0.37) ABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009130240-A1 ISOQUINOLINONE DERIVATIVES AS NK3 ANTAGONISTS H. LUNDBECK A/S (DK) 2009-10-29 WO claimed
WO-2009130240-A1 ISOQUINOLINONE DERIVATIVES AS NK3 ANTAGONISTS H. LUNDBECK A/S (DK) 2009-10-29 WO disclosed