SCHEMBL4319628

SCHEMBL4319628

N#Cc1cccc(-n2c(=S)[nH]c(N)c(N=O)c2=O)c1

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.40
NSD2 O96028 1/20 0.39
DRD2 P14416 1/20 0.37
DRD3 P35462 1/20 0.37
NOTUM Q6P988 1/20 0.37
CA12 O43570 6/20 0.37
CA1 P00915 6/20 0.37
CA2 P00918 6/20 0.37
CA9 Q16790 6/20 0.37
TDP2 O95551 1/20 0.36
GAA P10253 1/20 0.36
NOX4 Q9NPH5 1/20 0.35
XDH P47989 1/20 0.35
ALDH1A1 P00352 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ammonia Solution, Strong SCHEMBL4337843 0.84 ALOX5 (0.42) ALOX5NSD2DRD2DRD3NOTUM
SCHEMBL4499372 0.83 NSD2 (0.39) ALOX5NSD2DRD2DRD3NOTUM
SCHEMBL4492543 0.76 GAA (0.61) ALOX5NSD2DRD2DRD3NOTUM
SCHEMBL4316275 0.76 NSD2 (0.43) ALOX5NSD2DRD2DRD3NOTUM
SCHEMBL4489173 0.75 NSD2 (0.42) ALOX5NSD2DRD2DRD3NOTUM
SCHEMBL9954597 0.71 CA12 (0.64) CA12CA1CA2CA9ALDH1A1
SCHEMBL4456420 0.68 MPO (0.42) ALOX5NSD2DRD2DRD3TDP2
SCHEMBL1943938 0.67 MEN1 (0.43) GAAALDH1A1
SCHEMBL4501815 0.65 MEN1 (0.47) CA12CA1CA2CA9GAA
SCHEMBL7691283 0.64 GAA (0.39) GAAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010534-A1 THIOXANTHINE DERIVATIVES AND THEIR USE AS INHIBITORS OF MPO AstraZeneca AB (SE) 2009-01-07 EP disclosed
WO-2007120097-A1 THIOXANTHINE DERIVATIVES AND THEIR USE AS INHIBITORS OF MPO ASTRAZENECA AB (SE) 2007-10-25 WO disclosed