SCHEMBL4320876

SCHEMBL4320876

Oc1cc(O)c(Br)c(O)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 2/20 0.47
NQO1 P15559 1/20 0.43
TDP1 Q9NUW8 1/20 0.41
MEN1 O00255 2/20 0.39
CYP3A4 P08684 2/20 0.39
KMT2A Q03164 2/20 0.39
HPGD P15428 1/20 0.39
PTPN1 P18031 2/20 0.39
FASN P49327 1/20 0.38
CA1 P00915 2/20 0.36
CA2 P00918 1/20 0.36
CA4 P22748 1/20 0.36
CA6 P23280 1/20 0.36
NQO2 P16083 1/20 0.36
ALOX15 P16050 2/20 0.35
ALDH1A1 P00352 1/20 0.35
CA12 O43570 1/20 0.35
CA9 Q16790 1/20 0.35
PTGS1 P23219 1/20 0.35
DRD3 P35462 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23602095 0.80 CYP3A4 (0.46) BACE1TDP1MEN1CYP3A4KMT2A
SCHEMBL30279766 0.80 CYP3A4 (0.46) BACE1TDP1MEN1CYP3A4KMT2A
SCHEMBL4691914 0.80 TAAR1 (0.39) BACE1NQO1TDP1MEN1CYP3A4
SCHEMBL31167142 0.80 TAAR1 (0.39) BACE1NQO1TDP1MEN1CYP3A4
SCHEMBL7520723 0.79 CYP3A4 (0.47) TDP1CYP3A4HPGDPTPN1CA1
SCHEMBL515826 0.74 PTPN1 (0.52) BACE1TDP1CYP3A4HPGDPTPN1
SCHEMBL8763536 0.74 CA1 (0.50) TDP1MEN1CYP3A4KMT2AHPGD
SCHEMBL23628384 0.74 PTPN1 (0.44) MEN1CYP3A4KMT2AHPGDPTPN1
SCHEMBL21583494 0.73 HSD17B10 (0.50) TDP1MEN1CYP3A4KMT2AHPGD
SCHEMBL28794852 0.73 SELL (0.58) TDP1MEN1CYP3A4KMT2AHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113121965-A Insect pheromone-containing biodegradable agricultural film and preparation method thereof 陕西科技大学 2021-07-16 CN claimed
CN-109293493-B Novel benzhydryl compounds with mycobacterium tuberculosis inhibiting activity 清华大学 2021-08-03 CN disclosed
CN-113121965-A Insect pheromone-containing biodegradable agricultural film and preparation method thereof 陕西科技大学 2021-07-16 CN disclosed
CN-109293493-A With the inhibition active novel benzhydryl class compound of mycobacterium tuberculosis 清华大学 2019-02-01 CN disclosed
US-20090192152-A1 Novel Antigiardial Agents and Methods of Use Thereof UNIVERSITY OF MISSISSIPPI 2009-07-30 US disclosed
US-7468445-B2 Antigiardial agents and use thereof UNIVERSITY OF MISSISSIPPI (US) 2008-12-23 US disclosed
US-20060106091-A1 Antigiardial agents and use thereof THE UNIVERSITY OF MISSISSIPPI 2006-05-18 US disclosed
WO-2004014886-A1 ANTIGIARDIAL AGENTS AND USE THEREOF UNIVERSITY OF MISSISSIPPI (US) 2004-02-19 WO disclosed
US-5859067-A PREPARING BIS(2-HYDROXY-1-NAPHTHYL)DECANE FROM THE CORRESPONDING DIACID; FORMING ACID DICHLORIDE; TREATING WITH 2-NAPHTHOL; REARRANGEMENT; REDUCTION; INHIBITS ACTION OF ADENOSINE TRIPHOSPHATASE ROUFOGALIS BASIL DON (AU) 1999-01-12 US disclosed
US-5741821-A PHENOLIC ENZYME INHIBITORS THE UNIVERSITY OF SYDNEY (AU) 1998-04-21 US disclosed
EP-0703780-A4 USE OF NATURAL PRODUCTS AND RELATED SYNTHETIC COMPOUNDS FOR THE TREATMENT OF CARDIOVASCULAR DISEASE UNIV SYDNEY (AU) 1998-01-07 EP disclosed
EP-0703780-A1 USE OF NATURAL PRODUCTS AND RELATED SYNTHETIC COMPOUNDS FOR THE TREATMENT OF CARDIOVASCULAR DISEASE THE UNIVERSITY OF SYDNEY (AU) 1996-04-03 EP disclosed
WO-1994028886-A1 USE OF NATURAL PRODUCTS AND RELATED SYNTHETIC COMPOUNDS FOR THE TREATMENT OF CARDIOVASCULAR DISEASE THE UNIVERSITY OF SYDNEY (AU) 1994-12-22 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060106091-A1 Antigiardial agents and use thereof GPER1, ENPP2, ALPI BACE1 3168/4885NQO1 2161/4885TDP1 4344/4885
US-20090192152-A1 Novel Antigiardial Agents and Methods of Use Thereof ENPP2, GPER1, ALPI BACE1 3152/4885NQO1 2624/4885TDP1 4517/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.